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N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
9-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methanesulfonyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyrrolidine
4-(2-{1-[(5-chlorofuran-2-yl)methyl]piperidin-2-yl}ethyl)phenol
N-(3-phenylpropyl)-6-(pyridin-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-(5-chloro-2-methoxybenzenesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-1-(3-methoxybenzenesulfonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroquinolin-2-one
N-(2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]morpholin-2-yl}ethyl)methanesulfonamide
N-cyclopropyl-1-[(1s,4s)-4-[2-(4-chlorophenoxy)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl]benzoic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(pyridin-2-yl)acetamide
2-{9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
4-ethyl-3-[(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[(2-ethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
7-(3,6-dimethylpyrazin-2-yl)-4-(4-methyl-1H-imidazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1-acetylpiperidin-3-yl)-2,3,6-trimethylquinoline-4-carboxamide
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-N,N-diethylpiperidine-4-carboxamide
4-(3-fluorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]-1-[(3-methylphenyl)methyl]piperidin-2-one
4-fluoro-N-[(3R,5S)-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-3-yl]benzamide
1-{2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
3-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)sulfamoyl]dimethylamine
ethyl 4-(3-phenylpropyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine-4-carboxylate
4-methoxy-N-(2-methoxyethyl)-2-({1-[(3-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-[2-(ethylsulfanyl)phenyl]urea
(3aR,6aR)-2-(2-hydroxyethyl)-5-[3-(4-methoxyphenyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-7-(2-methoxyacetamido)-N,1-dimethyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-methylpropyl)piperidine-4-carboxamide
[(3R,4R)-1-(2-chloro-4,5-difluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]oxane-4-carboxamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,3-thiazole-4-carboxamide
N-(2-methoxyethyl)-1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-(5-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[1-(2,3-difluoro-4-methylbenzoyl)piperidin-4-yl]piperidin-3-ol
7-(2-cyclohexylethyl)-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-(4-fluorophenoxymethyl)-N-(1-methoxypropan-2-yl)-1,3-oxazole-4-carboxamide
2-{1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-methylformamido}-N,2-dimethylpropanamide
2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-(azepan-1-yl)-3-[4-chloro-2-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
8-(1H-indol-3-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[methyl(3-methylbutyl)carbamoyl]pyrrolidine-2-carboxylic acid
3-(3-methoxyphenyl)-N-[(2,3,4-trifluorophenyl)methyl]-1H-pyrazole-4-carboxamide
ethyl 4-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]piperidine-1-carboxylate