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N-[(5-methoxy-1H-indol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(azepan-1-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzonitrile
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-ethoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-methoxy-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-ethyl-3-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[2-(2-fluorophenyl)ethyl]-5-[1-(furan-3-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(4-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(3,4,5-trimethoxyphenyl)ethan-1-one
(3S,7S)-5-(2-ethoxybenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}amine
2-(3-methylbutyl)-8-(pyrrolidine-1-sulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S,5R)-4-[(cyclopropylmethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
2-(4-{6-azabicyclo[3.2.1]octane-6-carbonyl}piperidin-1-yl)-7-methanesulfonyl-4-methylquinazoline
1-{3-[4-(azetidin-1-ylmethyl)phenoxy]propyl}-1H-imidazole
N-(2-{[2-(phenylamino)pyrimidin-5-yl]formamido}ethyl)pyridine-3-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
3-{1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}propan-1-ol
(4aS,8aR)-6-(4-methyl-1H-imidazole-5-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(quinoline-6-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[2-(pyrrolidin-3-yl)benzoyl]piperidine
4-[5-(2-methoxypyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
(2R,6R)-4-[2-(morpholin-4-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}piperidin-3-ol
(3aR,6aS)-2-methyl-5-[2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
2-(2,4-difluorophenoxy)-1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}propan-1-one
4-hydroxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(3-methylphenyl)pyrimidine-5-carboxamide
5-(1-benzylpiperidin-4-yl)-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-(3-chloro-2,6-difluorophenyl)ethan-1-one
3-({1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[1-(pyrazin-2-yl)propan-2-yl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3aR,6aR)-2-[3-(2-fluorophenyl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol
4,6-dimethyl-2-(3-oxo-1,4-diazepan-1-yl)pyridine-3-carbonitrile
4-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]benzaldehyde
N-[2-(2-methylpropanesulfonyl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
4-[(2-acetamidoethyl)sulfamoyl]-N-(2-hydroxypropyl)benzamide
4-[({2-[(2-chloroprop-2-en-1-yl)oxy]-7-(methylsulfanyl)quinolin-3-yl}methyl)amino]adamantan-1-ol
5-chloro-2-(2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,6-dimethylpyrimidin-2-amine
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}urea
4-(5-ethylfuran-2-yl)-1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazole
[(3R,4R)-4-[(dimethylamino)methyl]-1-({4-[methyl(phenyl)amino]phenyl}methyl)pyrrolidin-3-yl]methanol
methyl 3-[(3S,4R)-1-[(3-fluorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
N-benzyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide