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N-(furan-2-ylmethyl)-3-[3-(1H-indol-3-yl)propanoyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N5-[(4-fluorophenyl)methyl]-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
naphthalen-1-yl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}methyl)-4-phenylbenzamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[(4-methoxyphenyl)methyl]urea
3-[(2-methoxyphenyl)methyl]-1-methyl-6-[(2-methyl-1,3-thiazol-5-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(4-fluorophenyl)-N-[(3R,5S)-5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]pyrrolidin-3-yl]acetamide
(3ar,6ar)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-[1-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-[3-(1-methoxyethyl)phenyl]-N,N-dimethylpyridine-3-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
2-{[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)amino}-N,N-dimethylpropanamide
2-methyl-1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(4-methylphenyl)piperazine
5-methyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[(2R,3R,6R)-5-(2,5-dimethylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(3aS,6aS)-2-[(3-chloro-2-fluorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(tert-butylsulfamoyl)-5-[(3-methylbutyl)amino]-N-[(1-methylpiperidin-3-yl)methyl]benzamide
4-[5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-2-one
4-(3,6-dimethylpyrazin-2-yl)-N-(quinolin-6-yl)piperazine-1-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-methoxypropan-1-one
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl]propanoate
1-(2-methylphenyl)-4-[3-(methylsulfanyl)propanoyl]piperazin-2-one
2-[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]-6-methylpyridine-3-carboxylic acid
2,3-dimethyl-7-[2-(1H-pyrrol-1-yl)acetyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(dimethylamino)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(4-fluorophenyl)-2-hydroxyethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
4-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-2-methylbutan-2-ol
N-cyclopropyl-4-{[3-(piperidin-1-yl)azetidin-1-yl]sulfonyl}benzamide
N-(carbamoylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
(3R,4R)-4-ethyl-1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]piperidine-3,4-diol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[1-methyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-yl]ethan-1-ol
1-(3-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
1'-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(2-cyclohexylethyl)-2-(1-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(3-cyclopentylpropyl)({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-[2-(3-aminopyrrolidin-1-yl)-2-oxoethyl]-1-benzyl-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-(2-ethoxyphenyl)-N'-[(4-methylphenyl)(pyridin-4-yl)methyl]propanediamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-8-methylimidazo[1,2-a]pyridine-2-carboxamide
3-propyl-5-{[2-(2,3,4-trifluorophenyl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
5-(1H-indol-1-ylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
(3aR,6aR)-2-(2-amino-6-methoxypyrimidin-4-yl)-5-ethyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2-dimethylpiperazine
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-N-methylpyridin-2-amine
8-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-[N-cycloheptyl-1-(3,5,7-trimethyl-1H-indol-2-yl)formamido]acetic acid