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7-methoxy-3-[2-(oxolan-3-yl)ethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
N,1-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-(4-chlorophenyl)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}butanamide
N-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1-methyl-1H-indole-6-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(pyrrolidin-1-yl)acetyl]-1,4-diazepan-5-one
2-(2,4-difluorophenoxy)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
6-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-(3-ethoxy-2-hydroxypropyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
methyl (2S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
4-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}thiomorpholine
1-[2-(4-methylpentyl)morpholin-4-yl]ethan-1-one
4-(2-fluoro-4-methoxyphenyl)-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole
2-(cyclopropylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
ethyl 4-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-amido)piperidine-1-carboxylate
(3S,4S)-3-hydroxy-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
(3aS,6aS)-N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
2-(2-aminoethyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)quinazolin-4-amine
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
5-methyl-5-(4-methylpent-3-en-1-yl)-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2H-chromen-2-one
2-(dimethylamino)-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-4-methylpyrimidine-5-carboxamide
2-methyl-4-[4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]but-3-yn-2-ol
2-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzoic acid
4-[hydroxy(pyridin-2-yl)methyl]-N-[2-(propan-2-ylsulfanyl)phenyl]piperidine-1-carboxamide
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)(oxan-2-ylmethyl)amine
N-(1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
1-cyclohexyl-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-2-yl}methanamine
(3S)-1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
2-{4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-indazol-3-yl)acetamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-1-[3-(1H-pyrazol-5-yl)phenyl]piperidine
{[3-(difluoromethoxy)phenyl]methyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(1,3-benzothiazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(1s,4s)-4-aminocyclohexyl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
5-methyl-1-(2-oxo-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{4-[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]piperazin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(2,4-difluorophenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
{3-[4-(2,3-dimethylphenyl)-1H-1,2,3-triazol-1-yl]propyl}(methyl)amine
2-[3-(1H-imidazol-1-yl)propyl]-N-(oxan-4-yl)-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-({7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
2-methyl-6-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)heptan-2-ol
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol