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2-(dimethyl-1,2-oxazol-4-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-tert-butyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-{2-[4-(dimethylamino)phenyl]acetyl}-1,4-diazepan-5-one
(3S,5R)-1-(1H-pyrrole-2-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3-thiadiazole-4-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
3-(hydroxymethyl)-N-(4-methoxy-3-propanamidophenyl)piperidine-1-carboxamide
(2R,3R)-3-{[2-(1H-pyrazol-1-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aS,7aR)-N-ethyl-4-[(5-methylfuran-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(4aR,8aS)-1-(5-methyl-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
[2-methoxy-5-(6-{[2-(morpholin-4-yl)ethyl]amino}pyridin-3-yl)phenyl]methanol
3-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-(2-methoxyethyl)-N-methylbenzamide
2-(2-phenylethyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-phenylpropyl)-1,4-diazepane
5-methyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}pyrimidin-2-amine
3-(1-methyl-1H-imidazol-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
1-[2-(benzyloxy)phenyl]-3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]urea
N,6-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-benzyl-3-[3-(4-hydroxypiperidin-1-yl)-3-oxopropyl]-1-methyl-2,3-dihydro-1H-indol-2-one
2-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-4-methoxyphenol
4-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-4-yl)pyridine
4-(2-fluoro-5-methylphenoxy)-1-[2-(5-oxopyrrolidin-2-yl)acetyl]piperidine-4-carboxylic acid
4-{4-[1-(2-methyl-1-benzofuran-7-yl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
1-(3-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(2,2-diphenylethyl)urea
7-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(2-methoxyphenyl)ethyl]-N-methylbenzamide
(1R,3S)-3-methoxy-7-(quinoline-6-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-{4-[6-(benzyloxy)pyridin-3-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetamide
3-(2-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(5-methylfuran-2-yl)benzamide
N-tert-butyl-3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
(2S)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-5-oxopyrrolidine-2-carboxamide
9-(3-chloro-2-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
2-cyclopentyl-8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2-methoxyphenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
4-ethyl-5-methyl-6-[4-(pyridin-4-ylmethyl)piperazin-1-yl]pyrimidin-2-amine
3-[3-({[(1S)-1-phenylpropyl]amino}methyl)-1H-indol-1-yl]propanamide
3-{[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
(2S,4R)-1-(1,4-dithiepan-6-yl)-N-methyl-4-[(pyrimidin-2-yl)amino]pyrrolidine-2-carboxamide
4-[(furan-2-ylmethyl)amino]-5-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 4-[(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
1-(4-methoxyphenyl)-3-(propan-2-yl)-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-ethyl-4-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]piperidine-1-carboxamide