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2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
1-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-oxopropyl}azepan-2-one
(1S,5R)-6-(1H-indole-6-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
(2S,3R)-3-hydroxy-2-({6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazol-3-yl}formamido)butanamide
1-methyl-4-(4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine
2-methyl-N-(1-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-methyl-5-{[(1R,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
N-methyl-2-[2-(1H-1,2,4-triazol-1-yl)propanamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]acetamide
methyl 4-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)butanoate
2-(5-{5H,6H,7H-cyclopenta[b]pyridin-3-yl}-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
6-[2-(2-methylpropyl)morpholin-4-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl]butane-1-sulfonamide
2-[(cyclohexylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-[(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
4-[5-(methoxymethyl)furan-2-carbonyl]-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-(cyclohexylmethyl)-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
3-{[2-(ethylamino)pyrimidin-5-yl]formamido}-3-(furan-2-yl)propanoic acid
2-{5-[(2-methoxyethoxy)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}-1H-1,3-benzodiazole
2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}acetamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
2,4-dimethyl-N-[4-(4-{[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-azaspiro[5.5]undecan-9-amine
5-cyclopropanecarbonyl-1'-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[4-(pyridin-2-yl)butyl]acetamide
3-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
2-{[(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N,N-dimethyl-2-[(2-methyl-6-propylpyrimidin-4-yl)amino]propanamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-phenylethyl)piperazine
2-(2-methylphenyl)-5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-thiazole
1-(5-chlorofuran-2-carbonyl)-3-(thiophene-2-carbonyl)piperidine
1-{2-methoxy-4-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
methyl (2S,4S)-4-(3-cyanobenzenesulfonamido)-1-methylpyrrolidine-2-carboxylate
2-[4-fluoro-2-(trifluoromethyl)phenyl]-N,N-dimethylpyridine-3-carboxamide
2-{1,3-dimethyl-4-[4-(pyrrolidin-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-ethyl-2-[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-indole
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-[2-(benzylsulfanyl)ethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(3-methoxyphenyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}propanamide
1-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
3-methyl-8-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,4-dihydroquinoxaline-2-carboxamide
4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}pyrimidine
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2,3,6-trifluorophenyl)methyl]amine