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2-(4-hydroxy-2-methylpyrimidine-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(6-chloro-2-methylquinoline-4-carbonyl)piperidin-3-amine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(3-fluorophenyl)methyl]piperidine-4-carboxamide
(2R,3R)-1'-(3-methylpyrazin-2-yl)-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-[4-(piperazin-1-yl)phenyl]pyrimidine
(3S,4S)-1-(5-chloropyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[2-(dimethylamino)ethyl]-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-N-methylpiperidin-3-amine
4-cyclobutanecarbonyl-9-(2,3-dihydro-1H-inden-1-yloxy)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
methyl (2S,4R)-1-methyl-4-[2-(propan-2-ylsulfanyl)acetamido]pyrrolidine-2-carboxylate
7-(cyclobutylmethyl)-6-oxo-N-(thiophen-2-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(furan-2-ylmethyl)piperidine-3-carboxamide
3-(2-{[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]amino}ethyl)-1,3-oxazolidin-2-one
3-cyclopentaneamido-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
N-cyclopropyl-4-{[1-(thiophen-3-yl)propan-2-yl]amino}pyridine-2-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(1H-pyrrole-2-carbonyl)piperazine
4-methyl-3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine
2-(dimethylamino)-N-ethyl-2-(3-fluorophenyl)-N-(2-hydroxyethyl)acetamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-(3-fluorophenyl)-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
7-[(4-fluorophenyl)methyl]-2-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-2,7-diazaspiro[4.5]decane
(4-{[1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-(3,4-dimethylphenyl)-N-[(2-methyl-1,3-thiazol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(hydroxymethyl)azepan-4-ol
N-cyclopentyl-1-methyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)azepane-2-carboxamide
1,6-dimethyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydroquinolin-4-one
4-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-2-methyl-1,2-dihydrophthalazin-1-one
(3aR,5S,6S,7aS)-2-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-isoindole-5,6-diol
3-(3-cyclohexyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)propanoic acid
(3S,4S)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
5-amino-3-[4-methoxy-3-(methoxymethyl)phenyl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
dimethyl[2-(2-{1-[4-(propan-2-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(2-methylphenyl)piperidine
8-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(cyclohex-1-en-1-ylmethyl)-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-(3-methylbutyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-chlorophenyl)-N-(5-hydroxypentyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
4-hydroxy-N-[2-(2-methoxyphenoxy)phenyl]piperidine-1-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-2-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2-dihydroquinoline-3-carboxamide
6-(benzyloxy)-4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(methylsulfanyl)-5-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}pyrimidine