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6-ethyl-N,2-dimethyl-N-(oxan-2-ylmethyl)quinoline-4-carboxamide
N-methyl-N-(piperidin-3-ylmethyl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
N-methyl-3-{[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
1-(2-methoxyphenyl)-3-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}urea
6-methyl-5-{5-[3-(morpholin-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})[2-(methylamino)ethyl]amine
3-chloro-N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
8-benzyl-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-{2-[(4-chlorophenyl)sulfanyl]acetyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[3-(4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}piperidin-1-yl)phenyl]pyridine-3-carboxamide
3-phenyl-N-(thiolan-3-yl)-1H-pyrazole-4-carboxamide
2-(methylamino)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidine-5-carboxamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
5-propyl-1'-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(3-cyclopentylpropyl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
1-(2-{[(3-hydroxypropyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
(4aS,8aR)-6-(2-amino-4-methylpyrimidine-5-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
2-(1-benzothiophen-3-yl)-2-(morpholin-4-yl)acetic acid
6-(cyclohex-1-ene-1-carbonyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(3-chloro-2-fluorobenzoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
6-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(benzenesulfonyl)methyl]-5-{spiro[2.3]hexan-1-yl}-1,2,4-oxadiazole
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopentylacetamide
{[3-({1-[3-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(1H-imidazol-2-ylmethyl)methylamine
8-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(4-{[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S,4R)-N,N-diethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-propanamidopyrrolidine-2-carboxamide
(2S,4S)-4-acetamido-N-ethyl-1-(8-fluoroquinoline-2-carbonyl)pyrrolidine-2-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-ol
1-{4-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-3-(piperidin-3-yl)benzamide
3-[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]pyrazine-2-carbonitrile
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-5-methyl-1,3,4-oxadiazole
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyphenyl)ethan-1-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
5-cyclopropyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,3,4-oxadiazol-2-amine
1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-3-phenylpyrrolidin-3-ol
N-(2-fluorophenyl)-3-({[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}amino)propanamide
6-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-[2-(dimethylsulfamoyl)ethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
3-(2-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
methyl 2-{2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}acetate