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N,N-dimethyl-5-{[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}furan-2-carboxamide
[(4-{[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
2-phenyl-1-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)ethan-1-ol
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(2-phenylethynyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-cyclopentyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(thiophen-3-ylmethyl)acetamide
7-(2-methoxyethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{2-chloro-5-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}furan-2-carboxamide
N-ethyl-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-(4-hydroxy-3-methoxyphenyl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(4aS,8aR)-1-(2-aminoethyl)-6-(3-phenoxypropanoyl)-decahydro-1,6-naphthyridin-2-one
8-(4-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(1-cyclohexyl-4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
6-[3-(furan-2-yl)benzoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[1-(4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}phenyl)ethyl]piperidine
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-[(3-methylphenyl)methyl]-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (1R,3S,3aR,6aS)-3-(5-ethylpyridin-2-yl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(3-methylpyridin-4-yl)piperazine
4-(6-chloro-1H-1,3-benzodiazol-2-yl)-2-ethoxyphenol
(1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-1-(2-phenylethyl)pyrrolidin-2-one
1-ethyl-3-{2-[(4-hydroxypiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-{[(1R,5S,8R)-8-(dimethylamino)-3-azabicyclo[3.2.1]octan-3-yl]methyl}benzoic acid
(4S)-3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenyl-1,3-oxazolidin-2-one
N-(1-methyl-1H-indazol-6-yl)-3-(pyridine-2-carbonyl)piperidine-1-carboxamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-(2,5-dimethoxyphenyl)-5,6-dimethylthieno[2,3-d]pyrimidine
8-(2,3-dihydroxybenzoyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
ethyl 1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopropane-1-carboxamide
2-ethyl-4-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]-1-(propan-2-yl)piperazine
N,N-dimethyl-3-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}sulfamoyl)benzamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
N-cyclobutyl-3-{[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]sulfonyl}benzamide
5-[(dimethylamino)methyl]-N-[2-(2-ethylphenoxy)ethyl]-N-methylfuran-2-carboxamide
(2S)-1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-N-ethylpyrrolidine-2-carboxamide
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(3-methylbut-2-en-1-yl)-1-(pyridine-2-carbonyl)piperidine-3-carboxylic acid
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-(pyrrolidine-1-carbonyl)-1,3-oxazole