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1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(1R,3S)-3-[1-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
3-(4-benzylpiperazine-1-carbonyl)-2-(cyclopentylmethyl)-1,6-dimethyl-1,4-dihydropyridin-4-one
(3aR,5R,6S,7aS)-2-[3-(2,5-dimethyl-1H-pyrrol-1-yl)-2-methylbenzoyl]-octahydro-1H-isoindole-5,6-diol
1-(5-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}-2-methylphenyl)imidazolidin-2-one
4-(quinolin-3-yl)pyridin-2-amine
1-[(3-methoxyphenyl)methyl]-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
1-{4-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
1-(2,5-dimethylfuran-3-carbonyl)-4-(1H-imidazol-2-yl)piperidine
2-{5-[1-(methoxymethyl)cyclobutyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}-6-methylpyridine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-cyclopentylpropanamide
5-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(4-chloro-2-fluorophenyl)-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3aS,6aR)-3-cyclopentyl-5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]pyridine-2-carbonitrile
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-methyl-4-[2-(methylamino)pyridine-3-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-[1-(7-chloro-4-methylquinolin-2-yl)pyrrolidin-3-yl]-N-methylacetamide
(3aR,6aR)-2-(oxane-4-carbonyl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(oxolan-2-ylmethyl)-5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine
(2S)-2-{2-[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]-1H-imidazol-1-yl}propanamide
N-ethyl-N-methyl-6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine-3-carboxamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N3-[2-(1H-indol-3-yl)ethyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(pyridin-3-ylmethyl)piperidin-3-amine
N,2,3-trimethyl-5-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-[2-(dimethylamino)-2,3-dihydro-1H-indene-2-carbonyl]-1,4-diazepan-5-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-{[1-(3-cyclopentylpropyl)piperidin-3-yl]methyl}-4-fluorobenzamide
N-(2-{[(3-methylphenyl)methyl]carbamoyl}phenyl)-1H-1,2,4-triazole-5-carboxamide
2-(4-cyclohexyl-3-oxopiperazin-1-yl)-2-(2-fluoro-3-methylphenyl)acetic acid
N-methyl-5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-({1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
methyl 3-(2-{[(2,4-dimethoxyphenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxylate
6-{[1-(2-chlorophenyl)piperidin-4-yl]amino}-2-methylheptan-2-ol
7-methyl-3-{[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)amino]methyl}quinolin-2-ol
(1R,5R)-6-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(4-hydroxyphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
4-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-1-methylpiperazine-2-carboxylic acid
2-(4-{[cyclopropyl(pyridin-4-ylmethyl)amino]methyl}phenyl)-6-(difluoromethyl)-3,4-dihydropyrimidin-4-one
N-{3-[2-(2-phenylethyl)morpholine-4-carbonyl]phenyl}acetamide
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-benzyl-4-[(2-butyl-1H-imidazol-4-yl)methyl]-1,4-diazepan-6-ol
2-[(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}phenyl)formamido]-N-methylacetamide
N-ethyl-3-[(2R)-2-hydroxy-2-phenylacetamido]-N-phenylbenzamide
3-(methylsulfanyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}propanamide
N-(2-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide