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4-methyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1,3-oxazole-5-carboxamide
(5R)-5-[1-(2-methoxyphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
ethyl 1-{4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanoyl}piperidine-2-carboxylate
(4aS,7aR)-1-{[3-(propan-2-yloxy)phenyl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,2-dimethyl-N-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
4-methyl-6-{[2-(trifluoromethyl)morpholin-4-yl]sulfonyl}quinolin-2-ol
4-(oxane-4-carbonyl)-2-(3-phenylpropyl)morpholine
2-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
1'-[4-(1H-pyrazol-3-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
N-(2-hydroxyethyl)-1-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-indole-4-carboxamide
2-(2-phenylethyl)-4-(thiophene-2-carbonyl)morpholine
N-({1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
2-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N,N,4-trimethyl-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-({1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
ethyl 4-({[3-(1,3-thiazol-4-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
(1-{1-[(3,5-difluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-(ethylamino)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
N-{[1-(methoxymethyl)cyclopropyl]methyl}-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(isoquinolin-5-ylmethyl)methylamine
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-(morpholin-4-ylmethyl)-N-[2-(2,4,6-trimethylphenoxy)ethyl]furan-3-carboxamide
3-(azepane-1-carbonyl)-N-[2-(1H-imidazol-1-yl)ethyl]benzene-1-sulfonamide
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(3,3,5,5-tetramethylcyclohexyl)propanamide
1-[benzyl(methyl)amino]-3-(5-{[(3-ethoxypropyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
N-[4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
2-(5-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
5-(4-methanesulfonylphenyl)pyrazin-2-amine
{3-ethyl-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}methanol
3-(4-hydroxyphenyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]propanamide
2-(2-hydroxyethyl)-9-(3-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1,2-oxazole-4-carboxamide
7-[(1-benzyl-1H-indol-6-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-({[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]amino}methyl)-5,8-dimethylquinolin-4-ol
[3-cyclopropanecarbonyl-9-(3-fluoropyridin-2-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-[3-(1H-indol-2-yl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
6-{[cyclopropyl(propyl)amino]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
1,3-dimethyl-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-(cyclopentylamino)-N-ethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)benzamide
4-(furan-2-ylmethyl)-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
N-[4-(3-methoxyphenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide