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1-[2-methyl-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]pyrrolidin-2-one
N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-chlorophenyl)methyl]-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
2-methyl-4-(4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenyl)butan-2-ol
2-methyl-6-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]pyrimidin-4-ol
3-(2-hydroxyphenyl)-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-{3-[(4-methoxyphenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}acetic acid
1-(2-methyl-4-{[2-methyl-2-(4-methylpiperidin-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-(2-methoxyethyl)-1-[1-(5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-3-(5-methylfuran-2-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
2,3,5-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
6-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methyl-1-[3-methyl-1-(4-methylquinolin-2-yl)-1H-pyrazol-5-yl]urea
methyl 5-[(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}acetamido)methyl]furan-2-carboxylate
N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
2,7-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(1-hydroxybutan-2-yl)-1-phenyl-N-(pyridin-2-ylmethyl)cyclopentane-1-carboxamide
2-(5-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N3-[2-(3-chlorophenyl)ethyl]-N5-cycloheptyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}benzoate
(furan-3-ylmethyl)(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
N-(1-{[5-(2-cyanophenyl)furan-2-yl]methyl}piperidin-4-yl)methanesulfonamide
(1R,5R)-6-[2-(4-fluorophenoxy)ethyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydroquinoxalin-2-one
3-methyl-1-propyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
1,1-dioxo-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1λ6-thiolane-3-carboxamide
4-fluorophenyl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N,5,6-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
[1-(7-fluoroquinazolin-4-yl)piperidin-4-yl](pyridin-2-yl)methanol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-propylpyrrolidin-3-yl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-6-(propan-2-yl)pyrimidin-2-amine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
N-[3-(methylsulfanyl)propyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-(4-hydroxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
(3aR,6aR)-2-[(3-chloro-4-methoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
methyl 4-(methylsulfanyl)-2-({5-[(quinolin-8-yloxy)methyl]-1,2-oxazol-3-yl}formamido)butanoate
(2-{2-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[3-(3-chlorophenyl)phenyl]-4-[(methylcarbamoyl)methyl]piperazine-1-carboxamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
9-[4-(dimethylamino)pyrimidin-2-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamido]-N,N-dimethylpropanamide
methyl 2-[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetate
3-(propan-2-yl)-5-[(2S)-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-2-yl]-1,2,4-oxadiazole