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2-(4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}morpholin-3-yl)acetic acid
(3S,4S)-4-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-1-(4-methoxybenzoyl)pyrrolidin-3-ol
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
1-{[2-(trifluoromethyl)phenyl]methyl}azepan-2-one
2,3-dimethyl-6-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-(methylsulfanyl)pyridine
N,2-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
N-(3,4-difluorophenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
N-methyl-4-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
N-[(1S,2R)-2-aminocyclobutyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
{1-[(2-chlorophenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
3-(2-phenylethyl)-8-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-2-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
2-methyl-4-(4-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(thiophene-3-carbonyl)piperidine
3-phenyl-5-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
5-(1,4-dioxane-2-carbonyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(3-methoxyphenyl)azetidin-1-yl]propan-1-one
[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
5-fluoro-2-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
(5S,9aS,9bS)-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
1,5-dimethyl-4-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
2-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]benzonitrile
2-methyl-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}quinoxaline
ethyl 1-[2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetyl]piperidine-2-carboxylate
4-fluoro-2-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenol
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N'1-methyl-N'1-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]cyclopropane-1,1-dicarboxamide
5-[({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
N-[2-(2,3-dimethoxyphenyl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-methoxy-5-methylphenyl)carbamoyl]piperidine-4-carboxylate
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-3-methylfuran-2-carboxamide
N-[2-(4-chlorophenoxy)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-ethylacetamide
6-(2,4-dimethylbenzoyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-N-(1-methyl-1H-indazol-5-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
4-[2-(ethylsulfanyl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-(4-hydroxybutan-2-yl)-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-2-one
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(1H-imidazol-1-yl)propyl]pyridin-2-amine
3-(3-methylbut-2-en-1-yl)-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidine-3-carboxylic acid
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
9-(6-aminopyrimidin-4-yl)-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-(trifluoromethyl)pyridine-3-carboxamide