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{2-[4-(propan-2-yloxy)phenyl]ethyl}({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-methylfuran-3-carboxamide
3-butyl-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
4-methoxy-3-({[1-(2-methoxyphenoxy)propan-2-yl]carbamoyl}amino)-N-methylbenzamide
1-(2H-1,3-benzodioxole-5-carbonyl)-2-(furan-2-yl)azepane
(4aS,7aR)-N-butyl-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N2-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(2S)-2-(methoxymethyl)-N-[4-(pyridin-3-yloxy)phenyl]pyrrolidine-1-carboxamide
1-(3,4-dimethylphenyl)-N-(1-ethylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-(2-methoxyethyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(pyridin-2-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-(furan-2-ylmethyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
1-[(4,5-dimethylfuran-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidine-3-carbonyl}pyridine
8-methyl-2-(morpholine-4-carbonyl)-2,8-diazaspiro[4.5]decane
4-(1-hydroxypropan-2-yl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1-butylpyrrolidin-3-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-(3-methylphenyl)-3-[1-(pyrrolidin-1-yl)ethyl]-4H-1,2,4-triazole
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
15-methyl-13-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-9-(pyridin-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
5-(methoxymethyl)-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
5-[(3,4-dimethoxyphenyl)methyl]-1-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-{[3-(benzyloxy)-4-methoxyphenyl]methyl}-3-(methoxymethyl)pyrrolidine
4-chloro-N,N-dimethyl-5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-1,3-thiazol-2-amine
8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
2-[4-(2-cyanophenyl)-3-oxopiperazin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
2-cyclopentyl-9-(2,6-dimethylpyrimidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(2-ethyl-3-oxopiperazin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidin-2-one
5-[(oxolan-2-ylmethoxy)methyl]-3-(thiophen-3-yl)-1,2,4-oxadiazole
N-[1-(pyrimidin-4-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-4-(4-fluorophenyl)butane-1,4-dione
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-(morpholin-4-yl)pyrimidine-5-carboxamide
1-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(4,6-dimethylpyrimidin-2-yl)methyl]benzamide
6-(cyclopropylmethoxy)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
[(1-cyclopentylpiperidin-4-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,2-oxazol-5-yl}methyl)-1H-1,3-benzodiazole
1-(2-{1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
ethyl 4-{[1-(1-methyl-1H-imidazol-2-yl)butyl]amino}piperidine-1-carboxylate
N-ethyl-1,3-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
ethyl 4-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperazine-1-carboxylate
3-(4-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile