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1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-methoxy-2-phenylethan-1-one
N-cyclopropyl-1-(2-methyl-4-phenylpyridine-3-carbonyl)piperazine-2-carboxamide
N-[(4-methoxyphenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2E)-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide
9-[3-(2-methoxyphenyl)propanoyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
4-{2-[(7-hydroxy-3,7-dimethyloctyl)amino]ethyl}-1-methylpiperidin-4-ol
N-[2-(1H-indol-3-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-phenylpiperidin-4-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-2-(2,4,6-trimethylphenyl)acetic acid
N5-ethyl-N3-methyl-N3-(naphthalen-1-ylmethyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4R)-4-methyl-3-(propan-2-yl)-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-ol
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(diethylamino)pyrrolidin-1-yl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propan-1-one
N-ethyl-4-(piperidin-3-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
9-(4-methoxypyrimidin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(azepan-1-yl)-3-[3-({[5-(morpholin-4-yl)pentyl]amino}methyl)phenoxy]propan-2-ol
(2E)-3-(2-chlorophenyl)-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
5-(2-phenylmorpholine-4-carbonyl)-1,3-benzothiazol-2-amine
N-{2-[({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)amino]ethyl}acetamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{4-[4-(trifluoromethyl)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
1-(2-fluorophenyl)-4-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}morpholine-2-carboxamide
1-[2-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
1-[(4-fluorophenyl)methyl]-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(propan-2-yl)-1,4-diazepane
5-[1-(benzenesulfonyl)cyclopropyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
ethyl 4-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
3-[(3R,4S)-1-(1H-indazole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-ol
6-(2-chlorophenyl)-2-(3-hydroxypiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(pyrazin-2-yl)propanamide
{2-oxo-2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethyl}urea
4-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1λ6-thiomorpholine-1,1-dione
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl](2-methoxyethyl)amine
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
methyl 1-[2-hydroxy-3-(3-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
4-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)piperazine-1-carboxamide
2-(4-fluorophenyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
(1R,5S,6S)-6-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
1-benzoyl-3-[2-(2,6-difluorophenyl)ethyl]piperidine
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]-4-(1H-pyrazol-1-yl)butanamide
2-methoxy-N-[1-methyl-5-(4-methyl-3-phenylpiperazine-1-carbonyl)-2-(pyridin-3-yl)-1H-1,3-benzodiazol-7-yl]acetamide
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-{5-[1-(4-chlorophenyl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-1,3-benzodiazole