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3-(1-methylpiperidin-3-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}propanamide
N-(3-hydroxybutyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[2-(3-acetylphenyl)-4-chlorophenyl]acetamide
3-[4-(4-methylphenyl)-2-[(pyrimidin-4-ylmethyl)amino]pyrimidin-5-yl]benzonitrile
9-hydroxy-3-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
(2S)-2,4-diamino-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)butanamide
1-(azocan-1-yl)-3-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
2-(2H-1,3-benzodioxol-5-yl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
1-cyclopentyl-5-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-hydroxypropanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[(thiophen-2-ylformamido)methyl]piperidine-1-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methanol
3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)thiomorpholine
(3aS,6aR)-5-(3-chloropyridin-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[3-(morpholin-4-yl)propyl]acetamide
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-4-yl)piperazine
1-(diphenylmethyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine
4-methyl-N-{2-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
1-[1'-(5-ethyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[4-(furan-2-yl)phenyl]-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
2-fluoro-N-methyl-5-sulfamoyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-[4-(1,3-benzoxazol-2-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[5-(1H-1,3-benzodiazol-2-yl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
2-methyl-N-(pyridin-2-ylmethyl)-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]aniline
(1S,5R)-3-methyl-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-[2-(dimethylamino)ethyl]-8-(2-ethoxypyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-ethyl-6-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
ethyl 4-{1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl}piperidine-1-carboxylate
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
2-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
1-methyl-3-[4-(4-{[(5-methylpyrazin-2-yl)methyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
6-[(diethylamino)methyl]-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
6-(pyrrolidine-1-carbonyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrazin-2-amine
6-methyl-1-(1,3-thiazol-4-ylmethyl)-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-(4H-1,2,4-triazol-3-ylmethyl)-4-[2-(trifluoromethyl)benzoyl]piperazine
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine