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3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
4-{1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-imidazol-2-yl}pyridine
6-ethyl-N-[(5-methylpyrazin-2-yl)methyl]-2-(morpholin-4-yl)pyrimidin-4-amine
4-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methylurea
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[2-(3-methylpyridin-2-yl)ethyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
9-(2-methoxypropanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methoxyphenyl)-1-methyl-3-{2-oxo-2-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}pyrrolidine-2,5-dione
2-hydroxy-3-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}butanamide
4-[2-(methylsulfanyl)pyrimidin-4-yl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]benzonitrile
1-[(1S,5R)-6-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyridine-3-carboxylic acid
1-(2-{1-[3-(4-methylphenyl)propanoyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-2-(trifluoromethyl)morpholine
N-{[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
1-(5,6,7-trimethoxy-3-{[(thiophen-3-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
(3R,9aR)-3-benzyl-8-(4-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-(oxan-4-ylmethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(3-hydroxypropyl)-9-[(4-methoxy-2,5-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
dimethyl({4-[1-(quinoline-8-carbonyl)piperidin-2-yl]phenyl}methyl)amine
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(2-methylquinolin-5-yl)urea
4-(4-fluoro-2-methylphenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
N-[(5-methoxy-1H-indol-2-yl)methyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
(1S,5R)-6-[4-(propan-2-yl)benzoyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}-2-(2-methylphenyl)pyridine
2-[5-(1-{[(4-chlorophenyl)methyl]sulfanyl}ethyl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-methylbutyl)-1H-pyrazole-3-carboxamide
2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)acetamide
1-(3-{2-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}phenyl)ethan-1-one
2-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-N-(2-methylpropyl)propanamide
4-(3-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}phenyl)morpholine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
5-(cycloheptylamino)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[methyl(phenyl)amino]propyl}-2-(pyridin-3-yl)acetamide
4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-[4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyrazin-2-ol
(2S,4S)-4-amino-N-methyl-1-(2-methyl-4-phenylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
2-methyl-7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(pyrazine-2-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-[(2,6-dimethoxyphenyl)methyl]-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(1-methyl-1H-imidazol-2-yl)-1H-pyrazol-4-yl]benzoic acid
methyl 4-({3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}amino)benzoate
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-methoxyphenyl)acetamide
1'-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one