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4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
4-(2-butyl-1H-imidazol-4-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2-aminopyridin-3-yl)methyl]-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[1-(4-methylpyridin-2-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
5-(2,3-dihydro-1H-inden-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[3-(2,4-dimethoxypyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(1S,4S)-2-(2-fluorophenyl)-5-[(2-methylphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(1R,5R)-6-[(1-ethyl-1H-indol-4-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
benzyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
6-cyclopentyl-3-{[(6-ethylpyrimidin-4-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{[3-(2-methylphenyl)piperidin-1-yl]methyl}pyridine
2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-[(2-methylphenyl)methyl]acetamide
2-[methyl(phenyl)amino]-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-[4-(4-chloro-3-fluorobenzoyl)-2-oxopiperazin-1-yl]benzonitrile
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}furan-3-carboxamide
ethyl 4-benzyl-1-[(8-methoxyquinolin-2-yl)methyl]piperidine-4-carboxylate
7-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[3-(3,4-difluorophenyl)phenyl]-1H-pyrazole
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3,4-dimethoxybenzamide
(4aS,8aR)-6-(2-ethoxybenzoyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
1-{3-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[2-(1H-pyrazol-1-yl)phenyl]urea
ethyl 3-(2-methoxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxylate
4-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
3-chloro-4-({1-[(4-chlorophenyl)methyl]piperidin-4-yl}oxy)-N-[2-(dimethylamino)ethyl]benzamide
2,2-dimethyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-ethyl-4-methyl-5-[1-(oxan-2-ylmethyl)-1H-imidazol-2-yl]-1H-imidazole
N-benzyl-5-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aR)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{2-[methyl(phenyl)amino]acetyl}-decahydro-2,7-naphthyridine-2-carboxamide
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-2-amine
2-[benzyl(methyl)amino]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one
5-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
(3S,4R)-1-(isoquinoline-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
ethyl 1-[2-(dimethylamino)ethyl]-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)-1λ6-thiolane-1,1-dione
4-({1-[(3-methoxyphenyl)carbamoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(4-pentanamidophenyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
3-[1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H-1,2,3-triazol-4-yl]piperidine
7-methyl-3-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(2,3,4-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1H-indole-2-carboxamide