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3-({4-[1-(4,4,4-trifluorobutyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
1-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-3-(3-methoxyphenoxy)propan-2-ol
7-(3,6-dimethylpyrazin-2-yl)-4-(morpholine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-methylbutyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
5-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1H-imidazole-4-carboxylic acid
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
4-benzyl-1-methyl-3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1-(propan-2-yl)piperidin-4-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methanesulfonamidoacetamide
3-{5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
8-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-methylpyridin-2-yl)methyl]pyridin-2-amine
1-[(6-methoxy-2H-chromen-3-yl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
3-[5-(5-fluoro-2-methoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(propan-2-yl)propanamide
N-(1,1-dioxo-1λ6-thian-4-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
4-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholine-2-carboxamide
1-({3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)azepan-2-one
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
3-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)urea
3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
5-chloro-2-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]pyrimidine
ethyl 4-(oxan-2-ylmethyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidine-4-carboxylate
(4aS,7aR)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-1-[2-(dimethylamino)ethyl]piperidin-2-one
2-[4-(hydroxymethyl)phenyl]-2-[4-(2-methoxyethoxy)piperidin-1-yl]acetic acid
2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
N-(2-methoxyethyl)-1-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-[1-(2,2-diphenylethyl)piperidin-4-yl]-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
5-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[4-(2,3-dihydro-1-benzofuran-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[2-hydroxy-3-(3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)propyl]piperidin-4-ol
[2,2-dimethyl-3-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)propyl]dimethylamine
N1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pentane-1,5-diamine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclohex-3-ene-1-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
methyl 4-{[(2-{1-[2-(3-fluorophenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-{3-azaspiro[5.5]undecan-9-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,2,2-trimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
2-(dimethylamino)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
1-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}piperidin-4-ol
(1S,5R)-3-(3-phenylpropyl)-6-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4S)-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3,3,4-trimethylpiperidin-4-ol
2-[2-({[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-cyclopropyl-N-[3-(2-oxopyrrolidin-1-yl)phenyl]-1H-pyrazole-5-carboxamide
N-(4-fluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
2-amino-6-(4-chlorophenyl)-4-(3,4-dihydroxyphenyl)pyridine-3-carbonitrile