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3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]piperidine
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
(2S)-2-amino-1-{6-methyl-5-[5-(3,3,3-trifluoropropyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}butan-1-one
3-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
5-(2-methoxy-2-methylpropanoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[2-({[2-(2-fluorophenyl)-2-hydroxyethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
ethyl({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-[2-(pyrrolidin-1-yl)ethyl]-1-(quinolin-7-yl)urea
2-hydroxy-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
5-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(4-{1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}phenyl)(methyl)amino]ethan-1-ol
{2-[1-(1H-imidazol-2-ylmethyl)piperidin-2-yl]ethyl}dimethylamine
3-[(3R,4S)-1-(2-methoxypyridine-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-cyclopropyl-9-(4-phenoxybutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1H-imidazol-2-ylmethyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
ethyl 4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-(2-hydroxyethyl)-5-(4-methylnaphthalene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
1-{5-[(3-cyclohexylpyrrolidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
1-[(4-fluorophenyl)methyl]-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1,4-diazepane
2-(3,4-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 4-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]carbamoyl}benzoate
3-(ethylsulfanyl)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-ethyl-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-3-carboxamide
N-ethyl-2-{4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]piperazin-1-yl}acetamide
2-[5-(ethoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
3-[6-(dimethylamino)pyridin-3-yl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-[7-(4-methyl-2-oxopentanoyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
8-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(ethylsulfanyl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}quinoline-2-carboxamide
2-[5-(7-chloro-4-methylquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-cyclopropyl-1-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]piperidine-3-carboxamide
N-{[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
2-(2-chlorophenyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 1-(thian-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
methyl[(4-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](2-phenylethyl)amine
5-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-1-azabicyclo[3.2.1]octane
3-ethyl-1-[(2,3,4-trifluorophenyl)methyl]piperidine-3-carboxylic acid
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
4-{1-[2-(morpholin-4-yl)-2-oxoethyl]piperidin-3-yl}benzoic acid
N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
ethyl 3-(2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
2-[3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)phenyl]-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
(3S,4S)-1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-propylpyrrolidine-3-carboxylic acid
N-ethyl-N-{[4-(propan-2-yl)phenyl]methyl}-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
{1-[(2,4,5-trimethoxyphenyl)methyl]azepan-2-yl}methanol
3-methoxy-N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide