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6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
methyl 2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]amino}benzoate
2-methyl-5-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
6-(2-chlorophenyl)-2-(2-ethylpyrrolidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[(2,3-difluorophenyl)methyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3R,4S)-1-(8-fluoroquinoline-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-amine
3-(2-{ethyl[(1-ethyl-1H-imidazol-2-yl)methyl]amino}-1-hydroxyethyl)phenol
2-methyl-5-{4-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-{1-methyl-5-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]-1H-pyrrol-3-yl}ethan-1-one
1-(2-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
3,4-difluoro-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
5-[(4-methylpiperazin-1-yl)methyl]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}furan-2-carboxamide
2-{4-[2-(pyridin-4-yl)acetyl]morpholin-3-yl}-1-(thiomorpholin-4-yl)ethan-1-one
5-fluoro-N4,N4-dimethyl-N2-[(4-methyl-1,3-benzoxazol-2-yl)methyl]pyrimidine-2,4-diamine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
1-(6-hydroxy-4-{[4-(2-phenylethoxy)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
3-methyl-1-(3-methylphenyl)-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}piperidine-4-carboxamide
(4aS,7aR)-4-acetyl-N-(2-chlorophenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2,3-dimethyl-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
2-(ethanesulfonyl)-1-(2-methoxyethyl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1H-imidazole
4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
5-[3-(4-fluorophenoxy)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-chloro-3-methyl-N-[(1-propylpiperidin-3-yl)methyl]benzamide
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}acetamide
3-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}-1,2-benzothiazole
N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-ethyl-1-(propan-2-yl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{methyl[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]amino}-1λ6-thiolane-1,1-dione
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-5-carboxamide
2-methyl-6-{1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-3-yl}pyrimidin-4-ol
1-[(4-chlorophenyl)methyl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
1,3-dimethyl-N-{1-oxaspiro[4.5]decan-3-yl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-(1-benzofuran-2-yl)-N-(furan-2-ylmethyl)-N-methyl-1,2,4-triazin-3-amine
4-tert-butyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
4-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-2,6-dimethylphenol
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-methyl-2-(morpholin-4-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-[4-(4-{[(3-fluoro-4-methoxyphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]quinoline-4-carboxylic acid
(1S,4R)-2-{[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
(4aS,8aR)-6-(1H-indole-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{[3-(furan-2-yl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
2-(2-methoxyphenoxy)-N-{[1-(propane-1-sulfonyl)piperidin-3-yl]methyl}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-hydroxy-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide