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N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-3-(pyridin-3-yl)propanamide
(1R,5R)-3-[(4-fluorophenyl)methanesulfonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(methoxymethyl)cyclopentyl]-1-(4-sulfamoylphenyl)urea
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(thian-4-yl)piperazine
1-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)piperidin-1-yl]ethan-1-one
N-(1,4-dithiepan-6-yl)-1-[(6-methylpyridin-2-yl)methyl]azepan-3-amine
(4aS,8aR)-1-(3-aminopropyl)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
3-[2-(ethylsulfanyl)ethyl]-1-(3-methoxyphenyl)urea
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pentane-1,2-dione
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(quinolin-5-ylmethyl)propanamide
3-[1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-3-yl]benzoic acid
8-benzyl-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-(4-{2-[(2,3-difluorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
5-{[methyl(thian-4-yl)amino]methyl}-N-(propan-2-yl)pyrimidin-2-amine
2-[4-(2-chloro-6-methylbenzenesulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-3-ethylpiperidine-3-carboxylic acid
2-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
N1,N1-dimethyl-N4-(2-phenoxyphenyl)piperazine-1,4-dicarboxamide
3-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3,9-diazaspiro[5.6]dodecan-10-one
1-(methoxymethyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]cyclopropane-1-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
4-[3-(hydroxymethyl)-7-methylquinolin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyrimidin-2-yl)-1,4-diazepane
9-methoxy-7-oxo-3-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[(2,6-difluorophenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-hydroxy-2-methyl-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
1-(2-chlorophenyl)-3-(1-{1-[2-(methylamino)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl)-1λ6-thiolane-1,1-dione
1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)azepan-4-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-phenoxyethan-1-one
N-methyl-2-(1-propylpiperidin-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2-dimethyl-3-[(pyridin-3-ylmethyl)amino]benzamide
1-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-cyclopropyl-2-[3-(3-methylphenyl)piperidin-1-yl]pyridine-4-carboxamide
2-{5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-(1-{[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}ethyl)hepta-1,6-dien-4-ol
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(1,3-thiazol-4-yl)acetamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(methylamino)pyridine-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide