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5-(1H-pyrazol-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)furan-2-sulfonamide
1-(3-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}propyl)piperidine-3-carboxamide
2-(2-phenyl-1H-imidazol-1-yl)-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
1-cyclopropyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
5-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2,4-dichlorophenoxy)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
1-(2-methoxyethyl)-4-[5-(3-methoxyphenyl)furan-2-carbonyl]piperazine
2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrazine
N,5-dimethyl-2-(2-methylpropanamido)-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]benzamide
2-(6-methoxynaphthalen-2-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]morpholine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-[3-({[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-(3-phenylpropyl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,3-benzoxazole
1-{2-amino-4-[(3-hydroxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(pyridin-2-yl)ethan-1-one
3-methyl-8-[2-(propan-2-yl)pyrimidin-4-yl]-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3H,4H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-4-(pyridin-3-yl)-1-(3,3,3-trifluoropropanesulfonyl)pyrrolidine-3-carboxylic acid
2-(4-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
3-(azepane-1-carbonyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R)-3-(dimethylamino)-1'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N4-cyclopropyl-6-(4-methoxy-2-methylphenyl)pyrimidine-2,4-diamine
6-methoxy-3-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-benzofuran-2-carboxamide
1-({1-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-ethyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-2-one
4-(2,3-dihydro-1H-inden-2-yl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
1-(1-benzofuran-5-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
3-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}benzonitrile
1-methyl-4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]piperazine
ethyl 1-[6,7-dimethoxy-3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)quinolin-2-yl]piperidine-3-carboxylate
N-(1,4-oxazepan-6-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamide
5-[(dimethyl-1,3-thiazol-4-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-(1H-imidazol-1-ylmethyl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-N-methylfuran-2-carboxamide
(1R,5S,6R)-3-[(2R)-2-hydroxy-2-phenylacetyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
(4aS,8aR)-6-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
1-cyclopentyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-(2-methoxy-5-methylphenyl)acetamide
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclobutan-1-amine
2-acetamido-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazole
N-[3-({[2-(dimethylamino)ethyl](oxolan-2-ylmethyl)carbamoyl}methoxy)phenyl]propanamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
2-(2-methylquinolin-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one