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1-ethyl-N-[2-(furan-2-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-[(1,3-thiazol-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3S,4R)-1-[4-(4-hydroxyphenyl)benzoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
2-methyl-1-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)-2-phenylpropan-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methoxyacetamide
methyl (2R,4S)-1-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-hydroxypiperidine-2-carboxylate
(3aS,6aS)-2-(2-methoxyethyl)-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-6-[3-(propan-2-yl)-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
(3aS,6aS)-2-cyclopentyl-5-[2-(3-methoxyphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
3-[(3R,4S)-1-[2-(4-fluoro-2-methylphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methoxypyridine-4-carboxamide
2-(benzyloxy)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-ethyl-4-methyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1,3-oxazole-5-carboxamide
2-(1-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
3-({[(2,5-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
(3S)-1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-N,N-dimethylpyrrolidin-3-amine
2-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperidine
3-[5-(3-phenoxypropanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-{3-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}ethan-1-one
ethyl 1-(2-methylpropyl)-5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3-(piperidin-3-yl)benzamide
1-[2-(morpholin-4-yl)ethyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N3-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
N-[2-(dimethylamino)ethyl]-3,5-dimethyl-N-[(2-methylphenyl)methyl]-1H-pyrrole-2-carboxamide
2-(3,4-dimethylphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
[2-(1,4-dimethylpiperazin-2-yl)ethyl](methyl)[(3-methylthiophen-2-yl)methyl]amine
2-methyl-4-(piperidin-3-yl)-6-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidine
2-cyclopentyl-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
[(3R,4R)-1-benzoyl-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-{[(1H-indazol-6-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N,N-dimethyl-4-({[4-(methylamino)pyrimidin-2-yl]amino}methyl)benzene-1-sulfonamide
2-ethyl-4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyrimidine
1-[(2-chloro-4-fluorophenyl)methyl]-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
N,N-dimethyl-5-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-methoxy-5-methylphenyl)-3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidine-1-carboxamide
N-(2-hydroxyethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(propan-2-yl)propanamide
N-cyclopropyl-3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propanamide
1-methyl-4-({[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)piperidin-4-ol
5-(3-acetylphenoxymethyl)-N-(furan-2-ylmethyl)-1H-pyrazole-3-carboxamide
1-(6-amino-2-methylpyrimidin-4-yl)-4-phenylpiperidin-4-ol
2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3,4-oxadiazole
N-[(4-phenyloxan-4-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
N,N-dimethyl-5-({4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine