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4-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1,3-thiazole-5-carboxamide
4-(piperidin-1-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
2-(carbamoylamino)-N-[(3R,4S)-1-[(3-chlorophenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
2-[methyl(2-phenylethyl)amino]-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(3S,4R)-1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-methylpropyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-4-sulfamoylbutanamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-(4-hydroxypiperidin-1-yl)-N-methylpyridine-3-carboxamide
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyridine-3-carboxamide
(1S,5R)-3-[2-(3-methoxyphenoxy)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
2-[(1S,5R)-6-[2-(benzenesulfonyl)ethyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-(3-hydroxy-3-methylbutyl)-N-[(2S)-1-hydroxybutan-2-yl]benzamide
5-[3-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-[(3R,4S)-4-cyclopropyl-1-(pyridazin-3-yl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylsulfanyl)acetamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-methylpyrazine
N-cyclopropyl-2-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
2-(cyclopent-2-en-1-yl)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
(2E)-1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
5-(2,2-diphenylethyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-(1-methyl-1H-pyrrole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-4-(1H-1,2,4-triazol-3-yl)benzamide
2-ethyl-5-{[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}pyrimidine
2-{[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
5-[(methylsulfanyl)methyl]-N-(quinolin-8-yl)furan-2-carboxamide
N-[1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
1-{[1-(morpholine-4-sulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-[(4-hydroxyquinazolin-2-yl)sulfanyl]-N-[1-(3-methylpyridin-2-yl)ethyl]acetamide
1-[2-(difluoromethoxy)benzoyl]-3-(2-ethylphenoxy)azetidine
3-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenol
N-[4-(2-methanesulfonylacetamido)phenyl]-5-methylfuran-2-carboxamide
N-(3-chloro-4-fluorophenyl)-6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
N-(butan-2-yl)-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-(dimethylamino)-7-(7-methyl-1-benzofuran-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-chlorophenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl (2R,4S)-4-hydroxy-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-2-carboxylate
2-{[(6-methoxypyridin-3-yl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
1-ethyl-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-{4-[ethyl(phenyl)carbamoyl]phenyl}-4-methyl-1,4-diazepane-1-carboxamide
(5S,9aS,9bS)-5-[4-(difluoromethoxy)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[4-methyl-5-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol