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1-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-(2-ethoxypyridin-3-yl)-3-(pyrrolidin-1-yl)pyrazine
1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)-3-(1,2,3-thiadiazol-5-yl)urea
4,4,4-trifluoro-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}butan-1-one
2-(adamantan-1-yl)-4-hydroxy-N-[3-(oxolan-3-yl)propyl]pyrimidine-5-carboxamide
2-chloro-N-[(2,6-dimethoxyphenyl)methyl]-5-acetamidobenzamide
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-indole
2-methyl-N-(1,2-oxazol-3-ylmethyl)-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1,6-dimethyl-N-[4-(methylamino)butyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(1-{3-[(pyridin-3-yl)amino]propyl}-1H-1,2,3-triazol-4-yl)phenol
2-amino-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(5-methylthiophene-2-carbonyl)piperidine
1-methyl-2-{5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-1,3-benzodiazole
1,3-dimethyl-5-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(4aS,8aR)-6-[3-(4-fluorophenyl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-(4,7-dimethylquinazolin-2-yl)-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
1'-(2-ethoxybenzoyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methoxyethoxy)ethan-1-one
N-[(4-fluoro-3-methylphenyl)methyl]oxane-2-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(dicyclopropylmethyl)methylamine
1-ethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-4-carboxamide
7-fluoro-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-methylquinoline-4-carboxamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(4aR,7aS)-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(2E)-3-phenylprop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(oxolan-2-ylmethyl)-8-[3-(pyridin-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N4-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-(2,3-dihydro-1H-indene-1-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-{[(3R,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2,4-dimethoxyphenyl)methyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
6-[(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]-1,4-oxazepan-6-ol
5-fluoro-2-({2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-3-methyl-1H-indole
1-phenyl-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
[(3-chloro-1-benzothiophen-2-yl)methyl]({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-2-(pyridin-3-yl)ethan-1-ol
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-3-(2-methylphenyl)propan-1-one
3-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-5-methoxy-1H-indazole
5-methyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]acetamide
5-(2-ethoxyethyl)-1-[(4-ethylphenyl)methyl]-3-methyl-1H-1,2,4-triazole
5-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclohexyl-N-[1-(1H-indol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
(isoquinolin-5-ylmethyl)(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-[4-(methylsulfanyl)phenyl]acetamide
(3R,4S)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine