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N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(pyrrolidin-1-yl)benzamide
4-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(4-fluorophenoxy)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-ol
N4-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(naphthalen-2-yloxy)propanamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}furan-2-carboxamide
2-(3-fluorophenyl)-N-({7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-[(2R,3R)-2-methoxy-1'-(pyridin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-methyl-4-{[5-(2-methyl-1-benzofuran-5-yl)-1,2,4-oxadiazol-3-yl]methyl}piperazine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-benzyl-N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-amine
2-(6-amino-5-methylpyridin-3-yl)benzonitrile
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-3-(4-fluorophenyl)benzamide
2-[4-methyl-3-(4-methylphenyl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
1-(3-oxo-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)pyrrolidin-2-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(1-methyl-1H-pyrazol-5-yl)-1H-pyrazol-1-yl]acetamide
({4-ethyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-({3-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]piperidin-1-yl}methyl)phenol
methyl 3-acetamido-6-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-yl)benzamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
8-(3-chloropyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(adamantan-1-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-3-carboxylic acid
8-[(2,4-dimethylphenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
1-ethyl-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-chloro-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,5R)-6-benzyl-3-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-chloro-6-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
1-(3-fluorophenyl)-3-(1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-phenyl-1-(3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
(3S,4R)-4-(2-methylphenyl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
6-[4-(3-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(1-benzothiophen-3-yl)-9-methoxy-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
6-methyl-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
3-{[(3-hydroxy-3-phenylpropyl)(methyl)amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-cyclohexyl-2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(3-methoxyphenyl)ethyl]propanamide
5-{[benzyl(methyl)amino]methyl}-N-(3-hydroxy-3-methylbutyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[3-(5-methylfuran-2-yl)butyl]-2,9-diazaspiro[5.5]undecan-3-one