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(4aR,7aS)-N,N-dimethyl-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-({2-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
N-(1-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
(3S,5R,9R)-5-hydroxy-11-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
3-[3-(5-methylfuran-2-yl)-5-(morpholin-4-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-({1-[6-(1-hydroxyethyl)pyridin-2-yl]piperidin-4-yl}methyl)acetamide
(3S,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
dimethyl({4-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)amine
2-phenyl-N-[(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-methoxy-1-methyl-1H-indole-2-carboxamide
ethyl 4-{[4-(3-methyl-4-oxopentanoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-(3-methoxyphenoxy)ethan-1-one
4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
1-(2-methoxyethyl)-N3-[2-(2-methoxyphenyl)ethyl]-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methanol
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(thiophene-3-sulfonyl)piperidin-3-yl]propanamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-N-[2-(propan-2-yloxy)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1,3-dimethyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2-fluorophenyl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propanamide
7-methoxy-3-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-[4-(azetidin-1-ylmethyl)phenoxy]-3-[benzyl(methyl)amino]propan-2-ol
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-(3-methoxypropyl)-1-[2-methyl-5-(1,2-oxazol-5-yl)benzenesulfonyl]piperidine
1-methyl-6-oxo-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(trimethylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-methyl-9-(3-methylbenzoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl 3-(furan-2-amido)-6-[(3-phenylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-methoxyphenyl)methyl]-N-propylpropanamide
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
(4aS,7aR)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-N-(3-methoxy-2,2-dimethylpropyl)thiophene-2-carboxamide
4-(carbamoylmethoxy)-N-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide
6-methoxy-3-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
3-phenyl-N-[(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]propanamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
2-(4-fluorophenyl)-N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-ol