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2-[(1-methylpiperidin-3-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
5-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
4-{[3-(dimethylamino)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
5-ethyl-2-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]pyrimidin-4-amine
3-[(phenylsulfanyl)methyl]-5-{pyrazolo[1,5-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S,4R)-4-(4-{2-[(5-fluoro-2-methylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-methoxy-6-(prop-2-en-1-yl)-4-[1-(1,3-thiazol-2-ylmethyl)-1H-imidazol-2-yl]phenol
N,N-dimethyl-4-({[6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
4-(4-methanesulfonylphenyl)-1-methyl-1H-pyrrolo[2,3-b]pyridine
3-ethyl-8-[(2-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
N-(2-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-2-yl}ethyl)acetamide
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-(piperazine-1-sulfonyl)benzamide
6-(benzyloxy)-1-cyclohexyl-4-(1H-imidazole-4-carbonyl)-1,4-diazepan-2-one
1-(cyclohexylmethyl)-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
methyl 4-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]benzoate
1-{3-[2-(4-chlorophenyl)morpholin-4-yl]-3-oxopropyl}azepan-2-one
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
3-chloro-N-cyclopentyl-4-({1-[1-(propan-2-yl)piperidin-4-yl]piperidin-4-yl}oxy)benzamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]morpholine-4-sulfonamide
2-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
6-(2,5-dimethylfuran-3-yl)-2-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[3-(2,4-dimethylphenoxy)propyl]-N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
(2E)-1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]-4-methylpent-2-en-1-one
N-butyl-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(oxane-4-carbonyl)piperidine
N-[1-(4-{[(4-phenyloxan-4-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
5-ethyl-1'-(4-ethyl-5-methylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(1H-imidazol-4-ylmethyl)-2-(4-methylpentyl)morpholine
3-(3-fluorophenyl)-N-(1H-indol-5-ylmethyl)-1H-pyrazole-4-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-amine
N-(5-chloro-2-methoxyphenyl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
3-[(cycloheptylamino)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
(2R,6R)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
{5-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-{2-[(5-ethylpyrimidin-2-yl)oxy]hex-5-en-1-yl}thiomorpholine
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[3-(trifluoromethyl)phenoxy]piperidine
2-(methylsulfanyl)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
(3S,4R)-1-(1H-indole-2-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-{[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
2-amino-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-butyl-N-(pyridin-3-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
2-[4-(adamantan-2-yl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol