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1-({[1-(3,5-dichlorophenyl)-2-hydroxyethyl]carbamoyl}methyl)piperidine-4-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(trimethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl[(2-methylfuran-3-yl)methyl]{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
5-(1H-imidazol-1-ylmethyl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)furan-2-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methoxypropan-1-one
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
2-methyl-7-oxo-N-[2-(3-phenylpiperidin-1-yl)ethyl]-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(thiophen-3-ylmethyl)piperidin-4-yl]propanamide
2-{1-[(4-methylphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-{[1-(3-hydroxypropyl)pyrrolidin-3-yl]methyl}benzoic acid
N-ethyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,3-dimethoxybenzamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
1-cyclopentanecarbonyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]piperidine-4-carboxamide
7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3,5-difluoropyridine-2-carboxamide
N-[(3R,4S)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-acetyl-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-{4-[3-(2,5-dioxoimidazolidin-4-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
(1S,4S)-2-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}-5-methyl-2,5-diazabicyclo[2.2.1]heptane
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)but-3-enamide
[(2S)-1-(4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
5-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyrazin-2-ol
4-{1-[3-(thiophen-2-yl)propanoyl]piperidin-3-yl}benzoic acid
1-(2-methyl-1,3-thiazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-phenyl-1,2,4-triazin-3-amine
6-[2-(2-chloro-4-methylphenoxy)ethyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
2-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-6-methylpyridine
1-(2-methylpropyl)-8-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
3-[(3-methoxypyrrolidin-1-yl)sulfonyl]-N-(1,3-thiazol-2-ylmethyl)benzamide
(4aR,7aS)-4-(3,5-dimethylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(2-hydroxyethyl)-8-[3-(pyridin-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(4aS,8aR)-6-(3,5-dichloropyridin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
2-(2,3-dimethylphenyl)-2-{4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-phenylbutan-1-one
(1S,5R)-6-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{[2-(furan-2-yl)azepan-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
2-{[(5-chloro-1-benzothiophen-3-yl)methyl]amino}-N-cyclopentylpropanamide
4-methyl-6-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-2-phenylpyrimidine
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-[(4-fluorophenyl)methyl]-5-[1-(3-methoxybenzoyl)piperidin-4-yl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
(1S,9aR)-1-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-octahydro-1H-quinolizine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(4-methoxyphenyl)-N-methylcyclopropane-1-carboxamide