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6-(benzyloxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-methoxy-N,1,2-trimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-indole-3-carboxamide
6-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N-ethyl-N-methylpyrimidin-4-amine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-6-methylphenol
ethyl 1-[(4-methoxyphenyl)methyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
4-acetyl-N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
methyl 3-{4-[2-(3-methoxyphenyl)acetyl]-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl}propanoate
1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-(3-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
N,N-dimethyl-3-[2-({[2-(pyrrolidin-1-yl)ethyl]carbamoyl}amino)phenyl]propanamide
1-(3-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)ethan-1-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(trifluoromethyl)benzene-1-sulfonamide
5-(2,4-difluorophenoxymethyl)-N-[2-(pyrazin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-acetyl-N-[3-(4-chlorophenyl)propyl]-1H-pyrazole-5-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
(2S)-1-(4-acetyl-4-phenylpiperidin-1-yl)-2-amino-3-(1H-imidazol-4-yl)propan-1-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}pyrrolidin-3-yl)benzoic acid
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
2-amino-7-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-4-(3-fluorophenyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
N-(4-fluoro-2-methylphenyl)-3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}propanamide
5-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-N-methylpyrimidin-2-amine
3-(1-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-1-oxopropan-2-yl)-3,4-dihydroquinazolin-4-one
2-cyclopropyl-8-[2-(2,3-dimethylphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(5-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}-2,3-dihydro-1-benzofuran-2-yl)methanamine
3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
N-benzyl-N-methyl-3-[1-(pyridine-3-sulfonyl)piperidin-4-yl]propanamide
6-chloro-3-fluoro-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
(4aR,8aS)-1-[3-(3-fluorophenyl)benzoyl]-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
(3aS,6aR)-5-(7-chloroquinolin-4-yl)-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3aS,6aS)-2-(cyclobutylmethyl)-5-(pyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-(1H-pyrazol-3-yl)benzamide
1-[3-(4-fluorophenoxy)propyl]-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
2-methyl-4-(3-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}phenyl)butan-2-ol
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-N,N-dimethylazepan-4-amine
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]-N-(1-phenylethyl)acetamide
(2S)-2-(morpholine-4-carbonyl)-N-[2-(propylsulfanyl)phenyl]pyrrolidine-1-carboxamide
1-{3-azaspiro[5.5]undecan-9-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-{1-[({[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2H-1,3-benzodioxole-5-carboxamide
6-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclopentyl-4-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
3-(4-hydroxycyclohexyl)-7,8-dimethyl-3,4-dihydroquinazolin-4-one
4-[(2S)-1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidine-2-carbonyl]morpholine