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(3R,4S)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-3,4-dimethylpiperidin-4-ol
1-(cyclohexylmethyl)-3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
(3R,4S)-4-propyl-1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-amine
1-[2-(oxolan-3-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-[5-(1-methyl-5-oxopyrrolidin-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methanesulfonylethan-1-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
1-(pyridin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{[4-(3-acetylphenyl)-5-(2-methyl-1,3-oxazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(2-ethoxyethyl)-3-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-5-carboxamide
5-(2-chlorophenyl)-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2-hydroxyethoxy)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
5-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(4-methoxyphenyl)methyl]-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
(1-{[1-(7-fluoro-4-methylquinolin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-methyl-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazole-5-carboxamide
6-chloro-2-methyl-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}quinoline-4-carboxamide
2-{imidazo[1,2-a]pyridin-2-ylformamido}-N-(2-methylphenyl)acetamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2-methylpropyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-chloro-N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-1H-indole-2-carboxamide
1-{2-[(1-methoxypropan-2-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidin-2-amine
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperazine-1-sulfonamide
4-(hydroxymethyl)-3-[(4-methylnaphthalen-1-yl)methyl]-1,3-oxazolidin-2-one
N-methyl-2-(methylamino)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
3-[(4-fluorophenyl)methyl]-5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(piperidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-[(2-ethylbutanamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
(1-methyl-1H-imidazol-2-yl)({1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl})methanol
1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl 6-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-3-(2-phenoxyacetamido)thieno[2,3-b]pyridine-2-carboxylate
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-ethyl-2,5-dimethyl-1H-pyrrole
N-[2-(3-fluorophenyl)ethyl]-5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
1-[4-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
N,2,3,5-tetramethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(6-methoxypyridazin-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
1-ethyl-4-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
2-[2,5-dioxo-4-(2-phenylethyl)-4-(piperidin-4-yl)imidazolidin-1-yl]-N-methylacetamide
3-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-phenylurea
N-[2-(4-methoxyphenyl)ethyl]-4-methyl-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide