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5-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecane-3-carbonyl]-1,2-oxazol-3-ol
ethyl 2-{[2-(2-phenylethyl)morpholine-4-carbonyl]amino}acetate
1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-{1-[2-(quinolin-8-yloxy)ethyl]-1H-imidazol-2-yl}benzonitrile
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(4-propanoylphenoxy)acetamide
ethyl 4-{3-[(cycloheptylamino)methyl]-6-methylquinolin-2-yl}piperazine-1-carboxylate
1-{4-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]thiophen-2-yl}ethan-1-one
5-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}pyridine-2,4-diol
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxylic acid
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[1-(4-methylbenzenesulfonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
1,3-dimethyl-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-1H-pyrazole-4-carboxamide
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
(2S,4S)-1-(2,2-diphenylethyl)-N-methyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]propanamide
(4aS,7aR)-4-(cyclopropylmethyl)-N-(3,5-dimethylphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-methyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazine-2-carboxylic acid
3-[(3-chloro-4-ethoxyphenyl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
ethyl 1-(cyclopropylmethyl)-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[2-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxamide
2-{2-[4-(dimethylcarbamoyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
[(2S,6S)-11-methoxy-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
4-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-1-(3-chlorophenyl)piperazin-2-one
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-[2-(diethylamino)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
(2S,3S)-2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-methylpentanamide
8-fluoro-2-({4-[(2-methoxyphenyl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
4-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
5-[4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
1-(4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-methyl-3-(2-phenylethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-5-carboxamide
2-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-cyclopropyl-6-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidine
1-methyl-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-[4-(trifluoromethoxy)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
4-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
(3R,4S)-4-{[(2,3-difluoro-6-methoxyphenyl)methyl](ethyl)amino}oxolan-3-ol
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-{3-[7-(1-hydroxy-2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
2-[4-(2-amino-4-phenylpyrimidine-5-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
(3S,9aR)-3-(4-aminobutyl)-8-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-ethoxyethyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
ethyl 2-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate