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6-methyl-5-(5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
(3aR,6aR)-2-(3-cyclopropylpropanoyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,2-dimethyl-2-(3-methylphenoxy)-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3-{2-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-methyl-2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
3-({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)-2,2-dimethylpropan-1-ol
(2E)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]butanamide
(3R,5S)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-ethyl-N,N-dimethyl-4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrrolidin-2-one
3-methyl-7-(4,7,8-trimethylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[4-(cyclopropylmethoxy)phenyl]-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(1H-indol-3-yl)ethyl]benzamide
1-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-[2-(methylamino)ethyl]pyrrolidin-2-one
(3aR,6aS)-5-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 4-benzyl-1-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxylate
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(4-methoxyphenyl)-3-phenylpropanamide
1-{[(2R,5S)-5-benzyloxolan-2-yl]methyl}piperidine-4-carboxylic acid
4-(2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethyl)morpholine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-amino-6-butanoyl-4-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
4-(2,4-dioxoimidazolidin-1-yl)-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]benzamide
3,5-dimethyl-4-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
2-[4-(1,4-oxazepan-4-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
5-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
6-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
1,2-dimethyl-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]acetamide
(3aS,6aS)-2-acetyl-5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{[(3-cyclopentylpropyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
(3E)-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}pent-3-en-1-one
1-[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
N-[(1R,3R)-3-aminocyclopentyl]-3-(2,3-dihydro-1H-indol-1-yl)propanamide
1-(furan-3-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}benzonitrile
2-tert-butyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-4-hydroxypyrimidine-5-carboxamide
7-cyclopropanecarbonyl-N-(2-phenoxyethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}thiophene-2-carboxamide
(3S,4S)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
3-(2-hydroxyphenyl)-N-[2-(methylsulfamoyl)ethyl]-1H-pyrazole-5-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide