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N-(cyclopent-3-en-1-yl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}-N-[2-(pyridin-2-yl)ethyl]thiophene-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(methoxymethyl)-N-methylfuran-2-carboxamide
N-(2-methoxyethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
8-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
5-butyl-1'-(4,6-dimethylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopropyl-5-oxo-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-3-carboxamide
methyl 5-[(2,2-dimethylpropyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidin-2-amine
3-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]benzonitrile
2-{[4-(5-ethyl-2-methylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3-hydroxy-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)naphthalen-2-ol
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-1-methyl-3-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-acetamido-4-fluorophenyl)-octahydropyrrolo[1,2-a]piperazine-2-carboxamide
3-{1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
N-ethyl-1-({4-[(6-methylpyridazin-3-yl)carbamoyl]phenyl}methyl)pyrrolidine-3-carboxamide
1-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-[(4-chlorophenyl)methyl]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
1-(2-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-fluoro-2-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-[(2R,4R,6S)-2-phenyl-6-[4-(propan-2-yl)phenyl]oxan-4-yl]acetamide
1-{2-methoxy-5-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
N4-(2-hydroxy-3-methoxypropyl)-N4-methyl-6-(propan-2-yl)pyrimidine-2,4-diamine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-(hydroxymethyl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-ol
methyl 4-{[(4-fluorophenyl)methyl](prop-2-en-1-yl)carbamoyl}butanoate
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(2-methoxyethyl)-N-methylbenzamide
benzyl 6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxylate
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-methyl-6-phenyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridazin-3-amine
ethyl 2-{1-[(3-cyanophenyl)methyl]piperidin-2-yl}acetate
N-(cyclopropylmethyl)-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
[(4-ethoxyphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
(2S,4S)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-[2-(3-methylphenyl)acetamido]pyrrolidine-2-carboxamide
ethyl 3-{[3-(phenylmethanesulfonamidomethyl)piperidine-1-carbonyl]amino}propanoate
5-[2-(6-hydroxy-1,4-oxazepan-4-yl)-2-oxoethyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 1-benzyl-3-cyclopropaneamido-5-{[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3,4-dimethoxyphenyl)methyl]-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[2-(piperidin-2-yl)ethyl]-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)acetic acid
2-({5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}thiophen-3-yl)acetamide
methyl 2-(2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
1-(2-aminoethyl)-N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide