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1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-(propan-2-yl)-1-[(1s,4s)-4-(2,4-dimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-amino-1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
ethyl 1-(2,4-dimethoxybenzoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(2S)-N2-ethyl-N1-[2-(4-methoxyphenyl)phenyl]pyrrolidine-1,2-dicarboxamide
5-(3-acetamidophenyl)furan-2-carboxylic acid
N-methyl-6-(pyridin-3-ylmethyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-(2,3-dihydro-1H-inden-2-yl)-3-methoxybenzamide
5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazole
(1R,5R)-N,N-dimethyl-6-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1,3-thiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methyl-N-[3-(3-methylpiperidin-1-yl)propyl]pyrimidin-2-amine
N-[(5-methylfuran-2-yl)methyl]-3-[1-(quinolin-8-ylmethyl)piperidin-3-yl]propanamide
(1S,9aR)-1-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)-octahydro-1H-quinolizine
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pent-4-en-1-one
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-methyl-7-[2-methyl-2-(morpholin-4-yl)propyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-chloro-N-[(3-methoxyphenyl)methyl]-1-methyl-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
(3S,4S)-1-(furan-3-ylmethyl)-4-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}pyrrolidin-3-ol
2-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)quinolin-4-ol
1-tert-butyl-4-[4-(2-phenylethyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-methylfuran-3-carboxamide
5-fluoro-2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(2,5-difluorophenyl)methyl]acetamide
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
[2-fluoro-5-(6-methoxypyridazin-3-yl)phenyl]methanol
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-4-fluoro-N-(oxolan-2-ylmethyl)benzamide
3-{[(5-methylthiophen-2-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
5-[4-(aminomethyl)piperidin-1-yl]-2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridine-2-carboxamide
N-cyclopropyl-1-(3-phenoxypropanoyl)piperazine-2-carboxamide
(3aR,6aS)-1-oxo-5-[(2-phenylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(1-ethyl-1H-indol-3-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{2-oxo-2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
(3S,4S)-1-[(8-fluoroquinolin-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[2-(2-ethoxyphenoxy)ethyl]piperidine-3-carboxamide
3-(3,4-difluorophenyl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
4-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1,4-oxazepane
2-(2,5-dimethoxyphenyl)-5-methyl-4-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-1,3-oxazole
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(2-methoxy-5-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methoxyphenyl)acetamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(pyridin-3-yloxy)propyl]acetamide
1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-(2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-2-carboxamide