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2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-(quinoxalin-6-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-{5-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
N-(furan-2-ylmethyl)-1-(hydroxymethyl)-9-methyl-3,9-diazaspiro[5.5]undecane-3-carboxamide
4-(2-methylpropyl)-6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidin-2-amine
3-[(3-acetamidopyrrolidin-1-yl)methyl]-N-(5-methyl-1,3-thiazol-2-yl)benzamide
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(quinoxalin-2-yl)-1H-pyrazol-1-yl]acetamide
1-(1,3-thiazol-2-yl)-1H-indazole-3-carboxylic acid
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N-[(2R,3R)-1'-[(3-ethoxy-4-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-methyl-4-oxo-1-(2-phenylethyl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
2-amino-6-(4-hydroxyphenyl)-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
1-cyclopentyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one
4-methoxy-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
7-cyclopropanecarbonyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
ethyl 1-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-2-carboxylate
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-5-methoxyphenol
[2-(1H-1,3-benzodiazol-2-yl)ethyl][1-(3-fluorophenyl)propan-2-yl]amine
[(3R,4R)-1-(3-chloro-2-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
8-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
N-{1-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}cyclohexanecarboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
2-{2,7-diazaspiro[4.5]decane-2-carbonyl}-N-propylaniline
4-(3-methylphenoxy)-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
1-[3-(5-methylfuran-2-yl)butyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(1H-imidazol-2-ylmethyl)methylamine
(3S,4R)-4-(3-fluorophenyl)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
(3R,4R)-4-(azepan-1-yl)-1-[(3-chloro-4,5-dimethoxyphenyl)methyl]piperidin-3-ol
(1S,5R)-3-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[5-(1,4-dioxane-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]pyrrolidine
(3S,4R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-methoxypiperidin-4-amine
N-[(2S,4R,6S)-2-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3-dimethylbutan-1-one
1-{2-[methyl({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]ethyl}piperidin-2-one
9-(3,5-difluorobenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}ethan-1-one
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
6-methoxy-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(hydroxymethyl)-1-[1-(pyridine-2-carbonyl)piperidine-4-carbonyl]piperidin-4-ol
3-[1-(1-ethyl-1H-indol-5-yl)-N-methylformamido]-N-methylbutanamide
2-{1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}pyridine
3-cyclopropyl-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazole
(3S,4R)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide