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N-[2-(3-methylthiophen-2-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
2-methyl-N-({4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}methyl)propanamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-(oxan-4-ylmethyl)benzamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
N5-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-oxobutanamide
1-({2-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[(4-methoxyphenyl)methyl]-1-methylurea
N-[2-(3-phenylpiperidin-1-yl)ethyl]oxane-4-carboxamide
3-methyl-4-[1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(prop-2-en-1-yl)-1H-pyrazole
2-(2-chlorophenyl)-3-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-[(thiophen-2-ylmethyl)amino]benzamide
6-{methyl[(5-methylfuran-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
[2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethyl]urea
N-[(5-chlorothiophen-2-yl)methyl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-[(1S,2R)-2-aminocyclobutyl]-3,3-diphenylpropanamide
5-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-4-(trifluoromethyl)pyrimidin-2-amine
1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}azetidin-3-ol
methyl 6-(2-phenylpropyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl}){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(3-phenylphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
(2R)-2-amino-N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-phenylacetamide
N-{3-[(2-methylpropyl)carbamoyl]phenyl}-2-(thiophen-2-yl)azetidine-1-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-1H-pyrazole-4-carboxamide
N-[(3S,4R)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
N-[3-(1H-imidazol-1-yl)propyl]-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[(3aS,6aS)-2-(3,5,7-trimethyl-1H-indole-2-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}acetamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylate
(3S,4S)-3-hydroxy-4-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-1λ6-thiolane-1,1-dione
2-(pyrrolidin-1-yl)-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyrimidin-4-amine
N-{[7-(5-acetylthiophen-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}-2,2-dimethylpropanamide
(1S,5R)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(oxane-4-carbonyl)pyrrolidin-3-yl]methanol
3-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)-3-(hydroxymethyl)pyrrolidin-3-ol
2-{3-[3-(quinoxalin-2-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
2-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
(3aS,6aS)-2-[(4-acetamidophenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid