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N-cyclopropyl-3-{5-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(5-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
5-(propan-2-yl)-3-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
2-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine-3-carbonyl)pyridine
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridine
7-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(4-fluorophenyl)-4-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]butane-1,4-dione
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
N-tert-butyl-2-methyl-3-[({2-[methyl(phenyl)amino]ethyl}carbamoyl)amino]benzamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(3S,4R)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
1-{4-[({[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}amino)methyl]phenyl}imidazolidin-2-one
N-(1,4-dioxan-2-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propanamide
1-ethyl-4-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
1-[(2,3-dimethoxyphenyl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
methyl 3-[({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)(oxolan-2-ylmethyl)sulfamoyl]thiophene-2-carboxylate
1-({1-benzyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyridin-2-one
5-(methoxymethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
[2-(1H-imidazol-1-yl)ethyl][(8-methoxyquinolin-2-yl)methyl]methylamine
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
2-chloro-5-(2-fluoro-6-methoxyphenyl)-N-methylbenzamide
2-(3-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}phenoxy)acetamide
methyl 3-{4-phenyl-5-[6-(trifluoromethyl)pyridin-3-yl]-1H-imidazol-1-yl}propanoate
1-{4-[5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
3-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
8-fluoro-N-[2-(2-oxoimidazolidin-1-yl)ethyl]quinoline-2-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylquinoline-6-carboxamide
3-ethyl-4-methyl-N-{[1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-(4-{2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyrazine
3-(1-methyl-1H-pyrrol-2-yl)-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(1H-pyrazol-3-ylmethyl)(pyridin-4-ylmethyl)amine
4-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}thiomorpholine
1-cyclopentyl-N-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-amine
methyl 6-[4-(2-phenoxyethyl)piperazin-1-yl]pyrimidine-4-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
6-fluoro-2-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]quinolin-4-ol
5-(4-fluoro-2-methoxyphenyl)pyrazin-2-amine
3-(6-chloro-2-methylpyridin-3-yl)-1-[(4,6-dimethylpyridin-2-yl)methyl]-1-methylurea
2-[(2,6-dichlorophenyl)methyl]-5-(piperidine-1-carbonyl)pyrimidin-4-ol
1-[2-methoxy-4-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,6-dimethoxypyridine-3-carboxamide
4-benzyl-1-(6-methyl-2-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
N-[4-(1H-pyrazol-1-yl)phenyl]-6-(pyridine-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide