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2-(1H-imidazol-2-yl)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
2-[2-(adamantan-1-yl)-N-methylacetamido]-2-(pyridin-3-yl)acetic acid
9-(2-hydroxy-3-methylbutanoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-(benzenesulfonyl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
{[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}(ethyl)methylamine
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
2-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
4-{[(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
2-({4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
3-[1-(2-methoxy-4-methylbenzenesulfonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
(3S,4R)-1-(1H-indazole-3-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-chloro-N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}thiophene-2-sulfonamide
3-(2-ethylbutyl)-8-[(2S)-2-(methylamino)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-4-(3-propylpyrrolidine-1-carbonyl)-1,3-oxazole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-phenylcyclopentane-1-carboxamide
5-{3-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
benzyl({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl})ethylamine
4-(5-chloropyridin-2-yl)-N-(1,3-dihydro-2-benzofuran-5-yl)piperazine-1-carboxamide
5-(1,2-oxazolidine-2-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
3-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}sulfonyl)benzonitrile
3-(4-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
4-{2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
N-{[2-(4-fluoro-2-methoxyphenyl)phenyl]methyl}propanamide
N-[3-(cyclohexylsulfanyl)propyl]-5-(methoxymethyl)furan-2-carboxamide
2,3,5-trimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]propan-1-one
N-{[(3S,4S)-1-[(4-ethynylphenyl)methyl]-3-hydroxypiperidin-4-yl]methyl}cyclopropanecarboxamide
3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-7-fluoro-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinolin-2-one
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}piperidine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methoxyphenyl)propanamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-ethyl-4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-2-one
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
2-[(1-methylpiperidin-2-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-({[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
1-cyclopentyl-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
5-methyl-1-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-fluoro-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-[5-benzyl-4-(2-methoxyacetyl)-2-oxopiperazin-1-yl]benzonitrile
4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
4-{[1-(3-cyclopropylpropanoyl)pyrrolidin-3-yl]methyl}benzoic acid
1-[(diethylcarbamoyl)methyl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(thiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine