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(2R,6R)-4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}-N-methylpyridin-2-amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
5-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-phenyl-3-(piperidin-3-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(methylsulfanyl)benzoyl]-N-(propan-2-yl)piperidine-1-carboxamide
5-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1-methyl-1H-1,2,3-benzotriazole
2-(2-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
8-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(morpholin-4-yl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propan-1-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidine
2-(ethylamino)-N,4-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-thiazole-5-carboxamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
1-({[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
(2S)-2-acetamido-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-(methylsulfanyl)butanamide
2,7-dioxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,3-diazepane-4-carboxamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-2-(pyridin-4-yl)acetamide
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
N-(furan-2-ylmethyl)-3-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
3-(2-fluorophenyl)-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-phenylacetamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(4-methoxyphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-2-carboxamide
1-{spiro[azepane-4,2'-chromene]-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{4-[(2,3-dihydroxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-pyrrol-1-yl)ethan-1-one
1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
1-(thiolan-3-yl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)-3-methylpyrazine
8-methoxy-5-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}quinoline
5-(3-cyano-6-methylpyridin-2-yl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({1-[(dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
3-[(3R,4S)-1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
methyl (1S,3S,3aR,6aS)-3-(furan-3-yl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-methyl-1,3-oxazole-4-carboxamide
4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}benzoic acid
7-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-methyl-1-oxopropan-2-yl)acetamide
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)thiophene-3-carboxamide
5,6-dimethyl-N-[2-(1H-1,2,4-triazol-1-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
(4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)methanamine
2-(1-ethylpiperidin-4-yl)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]acetamide
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl}){[5-(methoxymethyl)furan-2-yl]methyl}amine
1-({1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-1,4-diazepane
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-methyl-2-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide