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4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
3-[(3,3-dimethylcyclohexyl)amino]-N-(2-methoxyphenyl)propanamide
4-ethanesulfonamido-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
N-cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}propanamide
1-(2-aminoethyl)-N-(2,2-diphenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-benzyl-N,1-dimethyl-5-{spiro[indene-1,4'-piperidine]-1'-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-[4-({4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
1-(4-tert-butylphenyl)-N-(1-ethylpiperidin-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(naphthalen-1-yl)-N-[2-(pyrazin-2-yl)ethyl]-1,2,4-triazin-3-amine
(4aR,7aS)-1-(2-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
methyl 1-benzyl-3-cyclopropaneamido-5-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-hydroxyethyl)-5-(methoxymethyl)-N-(1,3-thiazol-2-ylmethyl)furan-2-carboxamide
5-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,3,4-oxadiazol-2-amine
1-[(4aR,8aS)-1-(2-methylbenzoyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
2-(dimethylamino)-N-(3,3-dimethylbutyl)-2-(4-methylphenyl)acetamide
1-{5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
5-({5-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
3-fluoro-4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzene-1-sulfonamide
(2S,3R)-2-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxybutan-1-one
1-(1,3-benzothiazol-2-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}piperidin-4-amine
methyl 3-{4-[1-(N-methyl-1-thiophen-3-ylformamido)-2-phenylethyl]piperidine-1-carbonyl}benzoate
2-[4-(hydroxymethyl)phenyl]-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
3-amino-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
2-methoxy-5-[2-(pyridin-4-yl)-1H-imidazol-1-yl]benzamide
2-(furan-2-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(dimethyl-1,2-oxazol-4-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
4-hydroxy-N-methyl-2-(pyridin-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
N-{[3-(cyclopentyloxy)phenyl]methyl}-3-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-2-methyl-4-(2-methylphenyl)piperazine
3-(1-butyl-1H-imidazol-2-yl)-1-(2-propoxybenzoyl)piperidine
N-(4,4-dimethylpentyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidine-4-carboxamide
N-(5-carbamoyl-2-methylphenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(propan-2-ylsulfanyl)acetamide
N-(1-{[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperidin-3-yl)acetamide
(4aS,8aR)-6-methanesulfonyl-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[4-(pyridin-3-yl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-(3-{[(4-chloro-2,6-dimethylphenyl)carbamoyl]amino}propyl)piperidine-3-carboxamide
N-butyl-2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-(2-ethoxyphenyl)-2-methylpyridine
2-(pyridin-2-yl)-7-[3-(pyridin-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-3-phenylpropanoic acid
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(pyridin-2-yl)propanoyl]piperidine-3-carboxylate
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-(2-fluorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine