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4-[(oxan-4-yl)sulfamoyl]-N-[(3S)-pyrrolidin-3-yl]benzamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,6-dimethyl-2-(morpholin-4-yl)pyrimidin-4-amine
3-cyclohexyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-pyrazole-4-carboxamide
4-[2-(4-fluorophenyl)ethyl]-11-(morpholin-4-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1,3-oxazole-4-carboxamide
2-{[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}acetamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-methylazepane-2-carboxamide
(3S,9aR)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-oxoethyl)-4-phenyl-1,2-dihydrophthalazin-1-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-8-sulfonamide
4-methylphenyl (7S,9aR)-7-(4-aminobutyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-(1H-imidazol-1-ylmethyl)-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridine
N-cyclohexyl-2-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]butanamide
N-[(2,3-dimethylphenyl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-fluoro-2-methylphenyl)methyl]piperidin-3-ol
5-[(2-chlorophenyl)methyl]-5-[1-(4-fluorobenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-{1-[(3-chloro-2,4-difluorophenyl)methyl]piperidin-4-yl}piperidin-4-ol
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-{2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]ethyl}benzamide
3-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]pyrrolidin-3-ol
N-[(3R,4R)-3-hydroxy-1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1,4-diazepan-1-yl]-4,6,7-trimethylquinazoline
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}propanamide
2-(dimethylamino)-N-[4-(3-hydroxy-4-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
N-[(4-fluorophenyl)methyl]-3-(2-hydroxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
7-(4-chlorophenyl)-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]propane-2-sulfonamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
9-[(1,5-dimethyl-1H-indol-2-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[(3R,4R)-4-(hydroxymethyl)-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
N,N-dimethyl-3-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
2-[1-(1H-indazole-3-carbonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
(3aR,6aR)-2-[(4-methoxypiperidin-1-yl)sulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-(2-methoxyethyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N,N-bis(prop-2-en-1-yl)piperidine-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
2-(2,3-difluorophenyl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
1-[3-({2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}amino)propyl]pyrrolidin-2-one
3-(3-fluorophenyl)-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(adamantan-2-ylmethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-(5-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridin-2-yl)methanesulfonamide