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N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
N-({5-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-ethyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
N-{5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetamido]-2-methylphenyl}-3-methylbenzamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(furan-2-ylmethyl)piperidine-2-carboxamide
ethyl 2-[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]acetate
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(3aS,7aR)-5-methyl-2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-(2-{2-[3-(2-methylphenyl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methyl-1H-pyrrole
2-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxyethyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(8-methyl-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}quinolin-3-yl)methanol
N-[2-(2-ethylphenoxy)ethyl]-2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]-N-methylacetamide
6-(2-aminoethyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-methylpyrimidin-4-amine
2-ethyl-9-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[3-(1-benzyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)propyl]pyrrolidin-2-one
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
6-(4-methoxyphenyl)-9-(quinoxaline-6-carbonyl)-6,9-diazaspiro[4.5]decan-7-one
4-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,4-oxazepane
ethyl 1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]piperidine-3-carboxylate
N-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[4-(isoquinolin-5-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-(5-fluoro-2-methylphenyl)-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,2,5-trimethyl-1,3-oxazole-4-carboxamide
2-(cyclopropylmethyl)-9-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[2-(2-chlorophenyl)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-(5,6,7,8-tetrahydroquinoxalin-5-yl)benzamide
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(methoxymethyl)piperidine
4-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-4-oxobutanamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[4-(propan-2-yloxy)benzoyl]pyrrolidin-3-yl]methanol
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)acetamide
6-cyclopentyl-1-methyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
6-(cyclopropylmethoxy)-4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-butyl-8-(2-ethoxyacetyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{5-[(3-methoxypyrrolidin-1-yl)methyl]thiophen-2-yl}-1H-pyrazole
4-benzyl-3-ethyl-1-[(1-methylpiperidin-4-yl)methyl]-1,4-diazepan-5-one
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
4-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-methyl-3-{3-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazol-3-yl]phenyl}pyrazine
5-methyl-2-(1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,3-benzodiazole
2-(methylsulfanyl)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}benzamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
2-{4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-yl}phenol
4-{[4-(2-aminoethyl)phenyl]methyl}-1-(2-methoxyphenyl)piperazin-2-one