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2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-4-yl)ethan-1-ol
5-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylpyrimidin-2-amine
1-methyl-4-[1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]piperazine
(1S,5R)-3-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]-1,3-thiazole
N-[3-(2-acetamido-3-methylbutanamido)phenyl]-3-methylbenzamide
6-(4-ethylphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
3-methyl-1-propyl-5-(thiophen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
methyl[(3-methyl-1H-pyrazol-5-yl)methyl][2-(2-methylpiperidin-1-yl)ethyl]amine
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-3-(4-methylphenyl)propan-1-one
1-(2-cyclohexylethyl)-3-hydroxy-3-({[(2-methoxyphenyl)methyl]amino}methyl)piperidin-2-one
benzyl N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}carbamate
4-(2-methyl-1H-imidazol-1-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine-4-carboxylic acid
2-(adamantan-1-yl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2,2-dimethyl-6-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3,4-dihydro-2H-pyran-4-one
ethyl 2-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
(9aR)-8-(3-methoxybenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-5-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]furan-2-carboxamide
6-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-ylmethyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-N-ethyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
4-{4-[1-(6-methoxypyridin-3-yl)-1H-imidazol-2-yl]phenyl}-2-methylbut-3-yn-2-ol
2-{2-[benzyl(methyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-[2-(2-phenoxyacetyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
5-chloro-2-[3-(2-hydroxypropan-2-yl)pyrrolidine-1-carbonyl]phenol
(1S,5R)-3-cyclobutanecarbonyl-6-(2-ethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-propyl-1,3-thiazole-4-carboxamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2-phenyl-1,3-oxazol-4-yl)methyl]amine
N-(3-hydroxypropyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-7-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
3-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
N-(2-hydroxy-3-phenoxypropyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}acetamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1-methoxypropan-2-yl)acetamide
2-(4-methoxy-3,5-dimethylphenyl)-2-{methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}acetic acid
7-methoxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(3-chlorophenyl)-4-(1H-imidazol-2-yl)-1-methyl-1H-pyrazole
N-[2-(oxan-2-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(5-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
3-(diphenylmethyl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-sulfonamide
4-ethyl-3-({1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-[4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-N-(propan-2-yl)acetamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]spiro[azepane-4,2'-chromene]
6-({[4-(aminomethyl)phenyl]methyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-[4-cyclohexyl-3-oxo-6-(pyridin-2-ylmethoxy)-1,4-diazepane-1-carbonyl]pyridin-1-ium-1-olate