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N-methyl-N-(oxolan-2-ylmethyl)-1-(propan-2-yl)piperidin-4-amine
2-{4-[(3-chloro-4,5-dimethoxyphenyl)methyl]piperazin-1-yl}-5-fluoropyrimidine
5-[3-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrimidine
8-(1-methoxypropan-2-yl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
7-[2-(4-chlorophenyl)morpholine-4-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-{1-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}benzoic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-3-carboxamide
methyl 3-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]carbamoyl}benzoate
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(propan-2-ylsulfanyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
4-[(furan-2-ylmethyl)amino]-N,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-fluoro-N2-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N2,N4,N4-trimethylpyrimidine-2,4-diamine
1-[(2,6-difluorophenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6,7-dimethoxy-2-[3-(pyrrolidin-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
4-(2-ethoxypyridine-3-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
(2R,6S)-4-{1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-4-yl}-2,6-dimethylmorpholine
N-[3-(1H-imidazol-1-yl)propyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
N-[(1-benzylpiperidin-3-yl)methyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-phenoxy-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-methoxy-1,2-dimethyl-1H-indole
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decane
2-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]-2-azaspiro[4.4]nonan-3-one
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-cyclopropyl-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine-4-carboxamide
8-[(2,3-dichlorophenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(3-methylpyridin-4-yl)methyl]benzamide
N-ethyl-7-methoxy-N-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7,8-dimethyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
(3S,4R)-1-(3,4-dimethoxybenzenesulfonyl)-4-(hydroxymethyl)piperidin-3-ol
N-methyl-N-(oxan-2-ylmethyl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
1-ethyl-4-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-(3,4-difluorophenyl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
3-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
4-[(2S,4R,6S)-6-benzyl-4-acetamidooxan-2-yl]benzoic acid
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4,6-dimethoxypyrimidin-2-yl)-2-(trifluoromethyl)morpholine
1-(2-methoxy-4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N,N,6-trimethyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-amino-3-ethyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-cyclopropyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,4-oxadiazol-2-amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[2-(morpholin-4-yl)benzoyl]piperidin-4-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethylpiperazine-1-carboxamide
N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
1-(carbamoylmethyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-N-(pyrimidin-4-ylmethyl)acetamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
2-(2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenoxy)-N,N-dimethylacetamide