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4-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
1-{4-[2-(3-fluorophenyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
2-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrazine
N-ethyl-2-(thiomorpholin-4-yl)pyridine-3-carboxamide
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,3-oxazole-4-carboxamide
3-ethyl-4-methyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
N-[(3R,4S)-1-(3-hydroxypropyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methanesulfonylpropanamide
1-(3-oxo-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propyl)azepan-2-one
1-{4-[2-(quinoxalin-2-yloxy)hex-5-en-1-yl]piperazin-1-yl}ethan-1-one
N5-(cyclohexylmethyl)-N3-methyl-4-oxo-1-(propan-2-yl)-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
2-(4-{[4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-2-(pyridin-2-yl)acetamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)propanamide
4-[5-(4-chloro-1,5-dimethyl-1H-pyrazol-3-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]pyridine
(2S,4R)-4-(dimethylamino)-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidine-2-carboxylic acid
2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}pyridine
N-[(2-fluorophenyl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-ethyl-2-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
4-(3-fluoro-4-methylbenzenesulfonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(3-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
N-{[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
1-(4-benzoylpiperazin-1-yl)-3-(4-hydroxyphenyl)propan-1-one
2-[2-(2,5-dimethylphenoxy)-N-methylpropanamido]acetic acid
(4aS,7aR)-1-(2-ethoxyacetyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
7-(2-methyl-5-propylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decane
6-[(3-fluorophenyl)methoxy]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
(2S)-2-[2-(6-ethoxypyridin-3-yl)-1H-imidazol-1-yl]propanamide
(3S,4S)-4-(4-fluorophenyl)-1-[(2-hydroxy-5-methylphenyl)methyl]piperidin-3-ol
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(4S)-4-phenyl-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,3-oxazolidin-2-one
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(4-methoxyphenyl)piperazine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(4-methylpyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
(2S,4S)-4-amino-1-(1-benzoylpiperidin-4-yl)-N-methylpyrrolidine-2-carboxamide
4-[(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}pyrrolidin-3-yl)methyl]benzoic acid
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
4-({7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N,N-dimethyl-5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carboxamide
4-benzyl-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(dimethylamino)ethyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine