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(3S)-1-(1,3-benzoxazol-2-yl)-N,N-dimethylazepan-3-amine
(dicyclopropylmethyl)({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyridin-3-yl)ethan-1-one
9-[(2-fluorophenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
[5-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)furan-2-yl]methanol
2-{4-[2-(3,4-difluorophenyl)ethyl]piperazin-1-yl}pyrazine
4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
(3S,4S)-4-(3-methoxyphenyl)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-ol
N-(2-hydroxyethyl)-N-methyl-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
(3S,9aR)-3-benzyl-8-(3-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-[2-(oxan-4-yl)ethyl]furan-2-carboxamide
3-methyl-7-(2-phenylquinolin-4-yl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-indol-2-yl)methanol
3-(methoxymethyl)-1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidine
4-methyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyridin-4-yl)pyrrolidin-3-yl]methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-methylphenyl)methyl]oxolane-3-carboxamide
N-(2-methoxyethyl)-4-[4-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
(2R)-2-hydroxy-3-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
(3R,4R)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-ethylpiperidine-3,4-diol
8-chloro-2-(furan-2-yl)-N-methyl-N-(oxan-4-yl)quinoline-4-carboxamide
(3aR,5S,6S,7aS)-2-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
N,N-dimethyl-4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-sulfonamide
N,4-dimethyl-5-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-[5-(2H-1,3-benzodioxol-5-yl)-3-ethyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-N-[2-(piperidin-1-yl)ethyl]pyridine-2-carboxamide
(3aR,5S,6S,7aS)-2-(4,7,8-trimethylquinolin-2-yl)-octahydro-1H-isoindole-5,6-diol
5-fluoro-2-(4-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrimidine
2-[2-(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethyl]pyridine
3-{[(methylcarbamoyl)(phenyl)methyl]sulfamoyl}-N-propylbenzamide
[(3S,5R)-1-(4,5-dimethylthiophene-2-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-[(4aR,8aR)-4a-hydroxy-7-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
3-({2-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
7-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]thiophene-2-carboxylate
4-({[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]amino}methyl)-1,2-dihydrophthalazin-1-one
(5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-methyl-1H-indol-2-yl)methanol
{4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]phenyl}methanol
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-(2-methoxy-5-phenylphenyl)acetamide
1-(2-aminoethyl)-N-(cyclohex-1-en-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2,3,6-trimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-2-(1,2-benzoxazol-3-yl)acetamide
(3S,5S,9R)-5-{[(3-fluorophenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
2-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
6-{[2-(pyridin-2-yl)pyrrolidin-1-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(1-{[3-(methylsulfanyl)phenyl]methyl}azetidin-3-yl)pyridine
5-fluoro-3-methyl-2-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-indole