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6-(benzyloxy)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-6-ethyl-2-methylquinoline
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
2-{1-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-imidazol-1-yl)ethan-1-one
9-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-methylpiperidine-2-carboxamide
2-(2-amino-6-fluoro-1,3-benzothiazol-4-yl)-N,N-bis(propan-2-yl)benzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-chloropyrimidin-2-amine
(2S)-3-hydroxy-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
4-[1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)piperidin-3-yl]morpholine
1-cyclopentanecarbonyl-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylfuran-2-carboxamide
N-(2-methoxyethyl)-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
4-(3-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1-methyl-1H-1,2,4-triazol-5-yl)morpholine
3-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
{4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
2-[(4-chlorophenyl)methyl]-8-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3,4-dimethoxyphenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpropanamide
4-{[5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-propyl-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-methyl-2-[3-(oxan-4-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
(2S)-1-(furan-2-ylmethyl)-N-[3-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
ethyl 1-[(2-hydroxy-4-methoxyphenyl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-ethyl-6-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidin-4-amine
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
3-methyl-6-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-1,2,3,4-tetrahydroquinazoline-2,4-dione
{2-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}dimethylamine
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(3S,9aR)-3-(4-aminobutyl)-8-[(3-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-({[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(1-{[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
4-ethyl-1-[(9-ethyl-9H-carbazol-3-yl)methyl]-1,4-diazepan-5-one
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-[(2-methylpropanamido)methyl]benzoate
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]sulfamoyl})amine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
4-fluoro-N-(2-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-(4-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
1-benzoyl-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazine
N-(2-methoxyethyl)-3-methyl-4-({[2-(pyridin-4-yl)ethyl]carbamoyl}amino)benzamide
4-[(dipropylamino)methyl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]benzamide
2-(4-methoxyphenyl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-({2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}methyl)benzoic acid
2-[5-(2,3-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 1-methoxy-2-oxo-8-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(3R,4S)-1-(5-methyl-1,3,4-thiadiazol-2-yl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
6-fluoro-2-[({1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)methyl]quinolin-4-ol