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1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-(furan-2-yl)propan-1-one
ethyl 4-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(pyridin-4-yl)propanamide
3-[1-(propane-2-sulfonyl)piperidin-3-yl]benzoic acid
N3-ethyl-N1-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}pyrrolidine-1,3-dicarboxamide
N-{[3-(benzyloxy)phenyl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
[(3R,4R)-1-(3,4-dimethylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N,N-dimethyl-3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazin-2-amine
7-methyl-3-[(5-methyl-1,2-oxazol-3-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)-1,2,5-thiadiazole-3-carboxamide
3-{[(4-fluorophenyl)methyl]amino}-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(1-methylpyrrolidin-2-yl)acetamide
N-[(3R,4R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-butyl-3-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)urea
9-(6-ethyl-2-methylpyrimidin-4-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(2-{[cyclopropyl(ethyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
5-{[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-1,2-dihydropyridin-2-one
6-(3-fluorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyridine-3-carboxamide
7-(2-methoxyethyl)-2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-butanamido-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide
N-(4-butanamido-3-methoxyphenyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-{1-[3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-2-yl}pyridine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-{1-methyl-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-2-yl}ethan-1-ol
3-(2-methoxyphenyl)-N-[2-(pyrimidin-5-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-4-[4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(1-methanesulfonyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
1-[(2-fluorophenyl)methyl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-6-oxopiperidine-3-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
8-(2H-1,3-benzodioxol-5-ylmethyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
1-(4-chlorophenyl)-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclopropane-1-carboxamide
N-phenyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrimidin-2-amine
(4aR,8aS)-1-(pyridin-3-ylmethyl)-6-(1,2,5-thiadiazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-{5-[(2S)-azetidine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1H-1,3-benzodiazol-1-yl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
ethyl 5-[({3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1,2-oxazol-5-yl}formamido)methyl]furan-2-carboxylate
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
ethyl 3-benzyl-1-(1H-indole-5-carbonyl)piperidine-3-carboxylate
1-cyclohexanecarbonyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)pyrrolidine-2-carboxamide
{3-[(3-chlorophenyl)methyl]-1-(9H-purin-6-yl)piperidin-3-yl}methanol
2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide